SCHEMBL20056636

SCHEMBL20056636

COc1ccc(Cl)cc1-c1ccc(O)c(C)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.53
TLR8 Q9NR97 2/20 0.51
ERN1 O75460 1/20 0.51
KCNMA1 Q12791 2/20 0.46
CXCL12 P48061 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 2/20 0.43
CTSA P10619 1/20 0.43
AGPAT2 O15120 2/20 0.42
SLC9A1 P19634 1/20 0.42
ABL1 P00519 1/20 0.42
AR P10275 1/20 0.42
WDR5 P61964 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20056401 0.83 ESR2 (0.46) ESR2TLR8CXCL12
SCHEMBL2410947 0.80 CA1 (0.61) ERN1KCNMA1ALDH1A1HPGDAR
SCHEMBL12834087 0.80 ERN1 (0.71) ERN1KCNMA1KMT2A
SCHEMBL20056483 0.79 ESR2 (0.57) ESR2TLR8MEN1KMT2A
SCHEMBL10093048 0.78 AGPAT2 (0.57) ERN1KCNMA1MEN1KMT2AALDH1A1
SCHEMBL14599496 0.78 HSD17B1 (0.52) ESR2TLR8MEN1KMT2AKDM4E
SCHEMBL20056607 0.78 KDM1A (0.52) TLR8CTSAAR
SCHEMBL18155551 0.76 TUBB4A (0.46) ERN1KCNMA1CXCL12MEN1KMT2A
SCHEMBL14499509 0.76 CYP1A2 (0.45) KDM4E
SCHEMBL7699644 0.75 ALDH1A1 (0.56) ERN1MEN1KMT2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970353-B1 MANNOSE DERIVATIVES FOR TREATING BACTERIAL INFECTIONS VERTEX PHARMA (US) 2018-04-18 EP disclosed