SCHEMBL20063089

SCHEMBL20063089

CC(C)c1cc(CO)cc(CO)n1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.38
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
HMGCR P04035 1/20 0.31
KDM5B Q9UGL1 1/20 0.31
RECQL P46063 1/20 0.31
EGLN2 Q96KS0 1/20 0.30
CCR1 P32246 1/20 0.30
SORD Q00796 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
TSHR P16473 1/20 0.30
CRHBP P24387 1/20 0.30
CYP2C19 P33261 1/20 0.30
CRHR2 Q13324 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20063090 0.80 NOS2 (0.52) NOS3NOS1NOS2CCR1
SCHEMBL18489341 0.80 NOS3 (0.38) ACHENOS3NOS1NOS2HMGCR
SCHEMBL4049194 0.80 NOS3 (0.34) NOS3NOS1NOS2CCR1CYP3A4
SCHEMBL4270536 0.78 ACHE (0.52) ACHERECQLCCR1TSHR
SCHEMBL15274618 0.76 NOS2 (0.38) NOS3NOS1NOS2KDM5BCCR1
SCHEMBL20063087 0.76 MAPT (0.35) ACHENOS3NOS1NOS2HMGCR
SCHEMBL3506786 0.74 HRH3 (0.42) NOS3NOS1NOS2
SCHEMBL20072601 0.72 ACHE (0.42) ACHENOS3NOS2KDM5BRECQL
SCHEMBL11030024 0.72 ACHE (0.42) ACHERECQLCCR1SORD
SCHEMBL5102672 0.72 RECQL (0.52) NOS3NOS1NOS2KDM5BRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180105508-A1 INHIBITORS OF PHOSPHOGLYCERATE DEHYDROGENASE (PHGDH) AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2018-04-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180105508-A1 INHIBITORS OF PHOSPHOGLYCERATE DEHYDROGENASE (PHGDH) AND USES THEREOF PHGDH, PGD, PGK1 ACHE 2915/4885NOS3 2532/4885NOS1 2516/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.