SCHEMBL2008249

SCHEMBL2008249

O=C(c1noc(-c2ccncn2)n1)c1c(Cl)n(Cc2ccc(Cl)cc2Cl)c2ccc(Cl)cc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.34
MAPT P10636 2/20 0.34
ALDH1A1 P00352 1/20 0.34
ALOX12 P18054 1/20 0.34
MAPK1 P28482 2/20 0.34
MAPK14 Q16539 1/20 0.34
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
VDR P11473 1/20 0.33
CYP2D6 P10635 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
CYP2C19 P33261 2/20 0.33
KDM4E B2RXH2 1/20 0.33
TSHR P16473 2/20 0.32
HIF1A Q16665 2/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006939 0.95 L3MBTL1 (0.37) LMNAMAPTALDH1A1ALOX12MAPK1
SCHEMBL2001504 0.94 FAAH (0.35) LMNAMAPTALDH1A1ALOX12MAPK1
SCHEMBL2008605 0.93 LMNA (0.41) LMNAMAPTALDH1A1ALOX12MAPK1
SCHEMBL2002620 0.92 PLA2G2A (0.37) LMNAMAPTALDH1A1MAPK1MEN1
SCHEMBL2002148 0.91 LMNA (0.34) LMNAMAPTMAPK14MEN1KMT2A
SCHEMBL2007854 0.91 FAAH (0.35) MAPTALDH1A1ALOX12MAPK14MEN1
SCHEMBL2005893 0.89 SCD (0.34) LMNAMAPTALDH1A1ALOX12MAPK1
SCHEMBL2004149 0.89 GRM5 (0.41) LMNAMAPTALDH1A1ALOX12VDR
SCHEMBL1999738 0.88 CYP2C9 (0.39) LMNAMAPTALDH1A1ALOX12MAPK1
SCHEMBL2003287 0.85 LMNA (0.34) LMNAMAPTALDH1A1ALOX12MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed