SCHEMBL2001504

SCHEMBL2001504

Cc1ccc2c(c1)c(C(=O)c1noc(-c3ccncn3)n1)c(Cl)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.35
MAPK14 Q16539 3/20 0.35
MAPK1 P28482 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
KDM4E B2RXH2 1/20 0.34
PTGS1 P23219 1/20 0.34
LMNA P02545 4/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TP53 P04637 2/20 0.32
CYP2C9 P11712 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MAPT P10636 1/20 0.32
ALOX12 P18054 1/20 0.32
P2RX7 Q99572 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2008249 0.94 LMNA (0.34) MAPK14MAPK1MEN1KMT2AKDM4E
SCHEMBL2006939 0.91 L3MBTL1 (0.37) MAPK14MAPK1MEN1KMT2AKDM4E
SCHEMBL2002486 0.91 FAAH (0.43) FAAHMAPK14MEN1KMT2APTGDR2
SCHEMBL2009499 0.90 FAAH (0.33) FAAHMAPK14MAPK1MEN1KMT2A
SCHEMBL2002620 0.90 PLA2G2A (0.37) MAPK1MEN1KMT2APTGDR2LMNA
SCHEMBL2003537 0.90 GRM5 (0.38) FAAHMAPK1MEN1KMT2APTGDR2
SCHEMBL2008605 0.90 LMNA (0.41) MAPK14MAPK1MEN1KMT2ALMNA
SCHEMBL2002148 0.89 LMNA (0.34) MAPK14MEN1KMT2ALMNASMN1; SMN2
SCHEMBL2004301 0.89 RAB9A (0.36) FAAHMAPK1MEN1KMT2APTGDR2
SCHEMBL2007239 0.87 TP53 (0.35) FAAHMAPK14MAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed