SCHEMBL2010345

SCHEMBL2010345

O=C(c1ncc(-c2ccncc2)o1)c1c(Cl)n(Cc2ccc(Cl)cc2)c2ccc(Cl)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
ALOX12 P18054 1/20 0.38
PPARG P37231 1/20 0.38
RECQL P46063 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ALOX5 P09917 1/20 0.37
ALOX5AP P20292 1/20 0.37
FAAH O00519 2/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
SRPK1 Q96SB4 1/20 0.34
IDO1 P14902 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1999528 0.94 ALOX5 (0.37) MEN1MAPTALOX15TSHRKMT2A
SCHEMBL2001753 0.93 FAAH (0.44) MEN1MAPTALOX15ALOX12KMT2A
SCHEMBL2005326 0.91 MEN1 (0.43) MEN1CYP3A4MAPTALOX15TSHR
SCHEMBL2008226 0.90 ALDH1A1 (0.41) MEN1CYP3A4KMT2AHDAC1HDAC6
SCHEMBL2005733 0.90 MEN1 (0.45) MEN1CYP3A4MAPTTSHRKMT2A
SCHEMBL2006262 0.90 CYP2C9 (0.40) CYP3A4MAPTTSHRALOX12KMT2A
SCHEMBL2000331 0.90 PTGES2 (0.41) MEN1CYP3A4MAPTALOX15TSHR
SCHEMBL2006132 0.90 ALOX5AP (0.43) MEN1CYP3A4MAPTTSHRKMT2A
SCHEMBL2004214 0.88 CCR9 (0.37) MEN1CYP3A4MAPTALOX15TSHR
SCHEMBL2003811 0.88 FAAH (0.41) MEN1CYP3A4MAPTALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed