SCHEMBL2006262

SCHEMBL2006262

O=C(c1ncc(-c2ccncc2)o1)c1c(Cl)n(Cc2ccc(Cl)cc2Cl)c2ccc(Cl)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.40
CYP3A4 P08684 2/20 0.40
TAAR1 Q96RJ0 1/20 0.36
LMNA P02545 3/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
ALOX12 P18054 1/20 0.36
CASP1 P29466 1/20 0.36
MAPK1 P28482 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
TSHR P16473 3/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
PMP22 Q01453 1/20 0.34
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003317 0.95 L3MBTL1 (0.38) CYP2C9CYP3A4TAAR1LMNAALDH1A1
SCHEMBL2006660 0.94 CYP2C9 (0.37) CYP2C9CYP3A4TAAR1LMNAALDH1A1
SCHEMBL2002674 0.93 LMNA (0.43) CYP2C9CYP3A4TAAR1LMNAALDH1A1
SCHEMBL2002487 0.92 LMNA (0.40) CYP2C9CYP3A4LMNAALDH1A1MAPT
SCHEMBL2004240 0.92 PLA2G2A (0.39) CYP2C9CYP3A4LMNAALDH1A1MAPT
SCHEMBL2005303 0.91 SLC26A4 (0.38) CYP2C9CYP3A4LMNAMAPTFAAH
SCHEMBL2009494 0.90 FAAH (0.37) CYP2C9CYP3A4LMNAALDH1A1MAPT
SCHEMBL2010345 0.90 MEN1 (0.38) CYP3A4LMNAMAPTALOX12MAPK1
SCHEMBL2006841 0.89 CYP3A4 (0.37) CYP2C9CYP3A4TAAR1LMNAALDH1A1
SCHEMBL2001356 0.89 FAAH (0.37) CYP2C9CYP3A4TAAR1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed