SCHEMBL20103607

SCHEMBL20103607

Cc1cc(OCc2nc3ccccc3n2C(=O)OC(C)(C)C)ccc1NC(=S)Nc1ccc(Cl)c(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 8/20 0.51
EPHX2 P34913 8/20 0.51
ALOX5AP P20292 1/20 0.51
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
ALDH1A1 P00352 2/20 0.41
PKM P14618 1/20 0.41
HTT P42858 2/20 0.40
LMNA P02545 1/20 0.40
THRB P10828 1/20 0.40
HPGD P15428 1/20 0.40
ALOX12 P18054 1/20 0.40
RAF1 P04049 1/20 0.39
MAPK3 P27361 1/20 0.39
NTRK1 P04629 1/20 0.39
NTRK2 Q16620 1/20 0.39
TP53 P04637 2/20 0.38
MAPT P10636 2/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20103613 0.91 ALOX5 (0.47) ALOX5EPHX2ALOX5APMEN1KMT2A
SCHEMBL20103477 0.84 EPHX2 (0.55) ALOX5EPHX2ALOX5APMEN1KMT2A
SCHEMBL20103604 0.82 ALOX5 (0.35) ALOX5EPHX2ALOX5APMEN1KMT2A
SCHEMBL20103615 0.75 NPC1 (0.56) ALOX5EPHX2MEN1KMT2AALDH1A1
SCHEMBL20103483 0.75 ALOX5 (0.53) ALOX5EPHX2ALOX5APMEN1KMT2A
SCHEMBL18711197 0.68 PPARG (0.40) MEN1KMT2ATP53MAPTRAB9A
SCHEMBL20103473 0.68 ALOX5 (0.67) ALOX5EPHX2ALOX5APMEN1KMT2A
SCHEMBL20103602 0.68 EPHX2 (1.00) ALOX5EPHX2ALOX5AP
SCHEMBL20103574 0.68 ALOX5 (0.67) ALOX5EPHX2ALOX5APMEN1KMT2A
SCHEMBL368032 0.67 CYP1A2 (0.45) MEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018077898-A1 N,N'-DIARYLUREA, N,N'-DIARYLTHIOUREA AND N,N'-DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE UNIVERSITÄT INNSBRUCK (AT) 2018-05-03 WO disclosed
EP-3315495-A1 N,N' -DIARYLUREA, N,N' -DIARYLTHIOUREA AND N,N' -DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE Universität Innsbruck (AT) 2018-05-02 EP disclosed