SCHEMBL20112979

SCHEMBL20112979

CC(C)CC1(C)OB(c2cc(F)c3c(c2)CC(=O)N3)OC1(C)C

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.32
GRIA1 P42261 1/20 0.30
CACNG8 Q8WXS5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25826937 0.89 ROCK1 (0.31) ROCK1
SCHEMBL20106736 0.88 GRIA1 (0.34) GRIA1CACNG8
SCHEMBL20112881 0.87 AHR (0.35)
SCHEMBL15288616 0.86 LIPG (0.40) ROCK1GRIA1CACNG8
SCHEMBL20112974 0.85 CSF1R (0.30)
SCHEMBL21493489 0.77 KIF11 (0.39) ROCK1
SCHEMBL20112906 0.75 LPL (0.31) GRIA1CACNG8
SCHEMBL18189371 0.72 LIPG (0.35) ROCK1
SCHEMBL18189401 0.72 GRIA1 (0.38) GRIA1CACNG8
SCHEMBL18189549 0.71 AHR (0.43) ROCK1GRIA1CACNG8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018080916-A1 FUSED AZAHETEROCYCLIC COMPOUNDS AND THEIR USE AS AMPA RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-03 WO disclosed