SCHEMBL20118406

SCHEMBL20118406

CCC1=NN(c2ccccc2)C(=O)[C@]12CC[C@H](NC(=O)c1cc(C)ccn1)CC2

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.44
SMYD3 Q9H7B4 1/20 0.42
GRM5 P41594 2/20 0.41
ACKR3 P25106 2/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
PDE4B Q07343 2/20 0.37
PDE4D Q08499 1/20 0.37
RIPK1 Q13546 1/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
ALDH1A1 P00352 1/20 0.37
USP30 Q70CQ3 1/20 0.36
BTK Q06187 2/20 0.36
CTSA P10619 1/20 0.36
NTRK1 P04629 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118174 0.82 CRHR1 (0.40) DHODHSMYD3GRM5ACKR3PDE4B
SCHEMBL20118167 0.75 SHMT2 (0.42) KDM4EALDH1A1MEN1KMT2A
SCHEMBL20118158 0.75 SHMT2 (0.42) KDM4EALDH1A1MEN1KMT2A
SCHEMBL20118157 0.73 SHMT2 (0.42) KDM4EALDH1A1MEN1KMT2A
SCHEMBL20118131 0.70 SHMT2 (0.46) KDM4EALDH1A1MEN1KMT2A
SCHEMBL20118216 0.69 L3MBTL1 (0.40) KDM4EHPGDHSD17B10ALDH1A1KMT2A
SCHEMBL20118195 0.68 HSD11B1 (0.44) PDE4BPDE4DRIPK1NTRK1
SCHEMBL20118414 0.67 TNKS (0.55) KDM4EHSD17B10
SCHEMBL20118215 0.67 ITGB1 (0.34) MEN1KMT2A
SCHEMBL20118187 0.65 PDE4B (0.41) CNR1CNR2PDE4BPDE4DHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed