SCHEMBL20118174

SCHEMBL20118174

CCC1=NN(c2ccc(F)cc2Cl)C(=O)[C@]12CC[C@H](NC(=O)c1cc(C)ccn1)CC2

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 3/20 0.40
CRHR2 Q13324 1/20 0.40
GRM5 P41594 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PDE4B Q07343 7/20 0.38
SMYD3 Q9H7B4 1/20 0.38
HPGD P15428 1/20 0.36
ACKR3 P25106 1/20 0.36
DHODH Q02127 2/20 0.36
MAPK14 Q16539 1/20 0.35
WDR5 P61964 1/20 0.34
ABL1 P00519 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118184 0.84 CRHR1 (0.39) CRHR1CRHR2MEN1KMT2APDE4B
SCHEMBL20118407 0.84 PDE4B (0.40) CRHR1CRHR2PDE4B
SCHEMBL20118406 0.82 DHODH (0.44) GRM5MEN1KMT2APDE4BSMYD3
SCHEMBL20118187 0.82 PDE4B (0.41) CRHR1CRHR2PDE4BHPGD
SCHEMBL20118213 0.82 LMNA (0.42) CRHR1CRHR2PDE4BHPGD
SCHEMBL20118188 0.80 KDM4E (0.47)
SCHEMBL20118191 0.79 CRHR1 (0.43) CRHR1CRHR2MEN1KMT2APDE4B
SCHEMBL20118169 0.79 P2RX7 (0.35) CRHR1CRHR2
SCHEMBL20118172 0.79 P2RX7 (0.35) CRHR1CRHR2
SCHEMBL20118047 0.79 RORC (0.43) CRHR1CRHR2MEN1KMT2APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed