SCHEMBL20118187

SCHEMBL20118187

CCC1=NN(c2ccc(F)cc2Cl)C(=O)[C@]12CC[C@H](NC(=O)c1cccc3cccnc13)CC2

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 7/20 0.41
TNKS O95271 3/20 0.41
TNKS2 Q9H2K2 3/20 0.41
CNR1 P21554 3/20 0.40
CNR2 P34972 3/20 0.40
CRHR1 P34998 3/20 0.40
CRHR2 Q13324 1/20 0.40
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
HPGD P15428 1/20 0.38
HSD11B1 P28845 1/20 0.38
PDE4D Q08499 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118213 0.91 LMNA (0.42) PDE4BTNKSTNKS2CRHR1CRHR2
SCHEMBL20118188 0.83 KDM4E (0.47) TNKS
SCHEMBL20118174 0.82 CRHR1 (0.40) PDE4BCRHR1CRHR2HPGD
SCHEMBL20118184 0.82 CRHR1 (0.39) PDE4BCRHR1CRHR2HPGD
SCHEMBL20118407 0.81 PDE4B (0.40) PDE4BCRHR1CRHR2
SCHEMBL20118132 0.81 LMNA (0.46) PDE4BTNKSTNKS2CRHR1CRHR2
SCHEMBL20118220 0.79 ALDH1A1 (0.50) PDE4BCRHR1CRHR2HPGDHSD11B1
SCHEMBL20118070 0.78 CRHR1 (0.42) PDE4BCNR1CNR2CRHR1CRHR2
SCHEMBL20118231 0.77 CRHR1 (0.37) CNR1CNR2CRHR1CRHR2HPGD
SCHEMBL20118172 0.77 P2RX7 (0.35) CRHR1CRHR2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed