SCHEMBL2012281

SCHEMBL2012281

Cc1ccc2c(c1)c(C(=O)c1cnc(-c3ccncc3)o1)c(Cl)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.38
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
LMNA P02545 3/20 0.36
KMT2A Q03164 3/20 0.36
TSHR P16473 2/20 0.36
MAPK1 P28482 2/20 0.36
MEN1 O00255 2/20 0.36
HTT P42858 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
MAPT P10636 2/20 0.35
ALDH1A1 P00352 2/20 0.35
ALOX12 P18054 1/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.35
PTGS1 P23219 1/20 0.35
TP53 P04637 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004625 0.94 CYP2C9 (0.40) CYP3A4CYP2C9LMNAKMT2ATSHR
SCHEMBL2008233 0.92 LMNA (0.39) FAAHCYP3A4CYP2C9LMNAKMT2A
SCHEMBL2001978 0.91 FAAH (0.45) FAAHCYP2C9KMT2AMEN1HTT
SCHEMBL1996791 0.91 PTGES2 (0.38) FAAHCYP3A4CYP2C9LMNAKMT2A
SCHEMBL2003297 0.91 L3MBTL1 (0.38) CYP3A4CYP2C9LMNAKMT2ATSHR
SCHEMBL2006426 0.90 LMNA (0.43) CYP3A4CYP2C9LMNAKMT2ATSHR
SCHEMBL2008195 0.90 FAAH (0.36) FAAHCYP3A4CYP2C9LMNAKMT2A
SCHEMBL2003542 0.90 MAPT (0.39) CYP3A4CYP2C9LMNAKMT2ATSHR
SCHEMBL2007905 0.90 FAAH (0.37) FAAHCYP3A4CYP2C9LMNAKMT2A
SCHEMBL2007346 0.89 ALOX5AP (0.39) CYP3A4CYP2C9LMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed