SCHEMBL20124031

SCHEMBL20124031

C=C1C(c2cccc(N)c2)=CCc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.42
HTR6 P50406 1/20 0.38
MAP4K4 O95819 2/20 0.37
MAPT P10636 4/20 0.37
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
LMNA P02545 2/20 0.37
HPGD P15428 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
MEN1 O00255 3/20 0.34
KMT2A Q03164 2/20 0.34
MECP2 P51608 1/20 0.34
TDP2 O95551 1/20 0.34
BRD4 O60885 2/20 0.33
PSIP1 O75475 1/20 0.33
AXL P30530 1/20 0.33
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20124017 0.80 TDP2 (0.32) MAOATDP2PRF1
SCHEMBL25985744 0.70 MAOA (0.54) MAOAMAP4K4MAPTALDH1A1KDM4E
SCHEMBL29471388 0.68 MAOA (0.68) MAOAMAP4K4MAPTALDH1A1KDM4E
SCHEMBL2023695 0.68 MAOA (0.68) MAOAMAP4K4MAPTALDH1A1KDM4E
SCHEMBL29700245 0.68 CHRNB4 (0.36) HTR6CYP3A4
SCHEMBL9329744 0.68 HSD17B1 (0.44) KDM4EMEN1KMT2ATDP2CYP3A4
SCHEMBL30643801 0.68 TP53 (0.37) ALDH1A1CYP3A4TSHR
SCHEMBL170839 0.67 ALDH1A1 (0.39) HTR6MAPTALDH1A1KDM4ELMNA
SCHEMBL29598333 0.67 ALDH1A1 (0.39) HTR6MAPTALDH1A1KDM4ELMNA
SCHEMBL2442271 0.66 MAOA (0.65) MAOAMAP4K4MAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2686298-B1 SUBSTITUTED DIPHENYL DERIVATIVES CREATIVE THERAPEUTICS GMBH (DE) 2018-05-09 EP disclosed