SCHEMBL2013334

SCHEMBL2013334

NCCc1ccc2ccccc2c1-c1cccc(F)c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.48
CYP1A1 P04798 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP1B1 Q16678 2/20 0.41
PRKDC P78527 1/20 0.41
ADORA2A P29274 1/20 0.40
DPP4 P27487 1/20 0.37
MPO P05164 2/20 0.37
SLC6A4 P31645 1/20 0.37
HTR2A P28223 2/20 0.36
TRPM8 Q7Z2W7 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
HPRT1 P00492 1/20 0.36
SYK P43405 1/20 0.36
HTR1A P08908 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2717827 0.88 TAAR1 (0.41) TAAR1CYP1A2MPOSLC6A4HTR2A
SCHEMBL2015662 0.82 CYP11B1 (0.38) TAAR1MPOSLC6A4HPRT1
SCHEMBL2012666 0.79 TAAR1 (0.47) TAAR1ADORA2AMPOSLC6A4HTR2A
SCHEMBL2011259 0.79 TAAR1 (0.43) TAAR1HTR2ASYKKMT2A
SCHEMBL28665841 0.74 ALOX5 (0.52) TAAR1CYP1A1CYP1A2CYP1B1PRKDC
SCHEMBL31331884 0.73 MPO (0.50) TAAR1CYP1A2MPOSLC6A4HTR2A
SCHEMBL17187823 0.73 MPO (0.50) TAAR1CYP1A2MPOSLC6A4HTR2A
SCHEMBL3906112 0.72 ADRA2C (0.60) TAAR1DPP4
Hydrochloric Acid SCHEMBL31331975 0.72 HTR1A (0.51) TAAR1CYP1A2MPOSLC6A4HTR2A
Hydrochloric Acid SCHEMBL20564378 0.72 TAAR1 (0.48) TAAR1CYP1A2MPOSLC6A4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed