SCHEMBL2013778

SCHEMBL2013778

CCC(=O)NC1CCN(c2c(CCN)cc(Cl)c3cccnc23)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.44
RAB9A P51151 5/20 0.44
ALOX12 P18054 5/20 0.44
L3MBTL1 Q9Y468 4/20 0.41
HTR5A P47898 1/20 0.41
MTNR1A P48039 4/20 0.40
MTNR1B P49286 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
MAPT P10636 1/20 0.40
MPI P34949 1/20 0.40
HTT P42858 1/20 0.40
SUV39H2 Q9H5I1 2/20 0.39
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
METAP2 P50579 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2013328 0.91 L3MBTL1 (0.45) NPC1RAB9AALOX12L3MBTL1MEN1
SCHEMBL2017715 0.89 MTNR1A (0.41) NPC1RAB9AALOX12L3MBTL1HTR5A
SCHEMBL2017265 0.85 NPC1 (0.48) NPC1RAB9AALOX12L3MBTL1HTR5A
SCHEMBL2017031 0.85 NPC1 (0.48) NPC1RAB9AALOX12L3MBTL1HTR5A
SCHEMBL2012926 0.85 SMO (0.48) NPC1RAB9AALOX12L3MBTL1HTR5A
SCHEMBL2013775 0.85 ALOX12 (0.50) NPC1RAB9AALOX12L3MBTL1MTNR1A
SCHEMBL2014688 0.84 NPC1 (0.37) NPC1RAB9AALOX12L3MBTL1HTR5A
SCHEMBL2011476 0.82 METAP2 (0.43) NPC1RAB9AALOX12L3MBTL1MEN1
SCHEMBL2011479 0.82 METAP2 (0.43) NPC1RAB9AALOX12L3MBTL1MEN1
SCHEMBL2015791 0.81 METAP2 (0.42) NPC1RAB9AALOX12L3MBTL1HTR5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed