SCHEMBL2014424

SCHEMBL2014424

C=C(C)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
NPFFR2 Q9Y5X5 1/20 0.50
SRD5A2 P31213 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GAA P10253 1/20 0.43
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
PKM P14618 1/20 0.42
RAB9A P51151 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HPGD P15428 3/20 0.42
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31599679 1.00 TSHR (0.52) TSHRNPFFR2SRD5A2MEN1KMT2A
SCHEMBL10336410 0.82 HSD17B10 (0.48) TSHRNPFFR2GAAHSD17B10HPGD
SCHEMBL30482512 0.82 MEN1 (0.38) TSHRNPFFR2SRD5A2MEN1KMT2A
SCHEMBL19153456 0.82 TSHR (0.45) TSHRNPFFR2KMT2ASMN1; SMN2GAA
SCHEMBL11145835 0.82 HSP90AA1 (0.49) TSHRNPFFR2SMN1; SMN2HSD17B10HPGD
SCHEMBL9274485 0.82 MEN1 (0.38) TSHRNPFFR2SRD5A2MEN1KMT2A
SCHEMBL6128400 0.82 CYP3A4 (0.45) MEN1KMT2AGAAKDM4ENPC1
SCHEMBL11012802 0.80 CYP3A4 (0.46) TSHRNPFFR2MEN1KMT2ASMN1; SMN2
SCHEMBL22775248 0.80 CA12 (0.48) TSHRNPFFR2MEN1KMT2ASMN1; SMN2
SCHEMBL7982038 0.80 MAOA (0.43) TSHRMEN1KMT2ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12404253-B2 2,4,6-trisubstituted 1,3,5-triazines as modulators of CX3CR1 ASTRAZENECA AB (SE) 2025-09-02 US disclosed
EP-4605388-A1 <SUP2/>? <SUB2/>?3?2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CXCR1 Astrazeneca AB (SE) 2025-08-27 EP disclosed
US-20240383866-A1 2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CX3CR1 ASTRAZENECA AB (SE) 2024-11-21 US disclosed
US-20240199558-A1 2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CX3CR1 ASTRAZENECA AB (SE) 2024-06-20 US disclosed
WO-2024083933-A1 2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CX 3CR1 ASTRAZENECA AB (SE) 2024-04-25 WO disclosed
US-20220179312-A1 PATTERN FORMING METHOD AND METHOD FOR MANUFACTURING ELECTRONIC DEVICE FUJIFILM CORPORATION (JP) 2022-06-09 US disclosed
US-9417530-B2 Method for developing resist, method for forming a resist pattern, method for producing a mold, and developing fluid utilized in these methods FUJIFILM CORPORATION (JP) 2016-08-16 US disclosed
US-20150008211-A1 METHOD FOR DEVELOPING RESIST, METHOD FOR FORMING A RESIST PATTERN, METHOD FOR PRODUCING A MOLD, AND DEVELOPING FLUID UTILIZED IN THESE METHODS FUJIFILM CORPORATION (JP) 2015-01-08 US disclosed
CN-102652159-B Stain-resistant aqueous coating composition AKZO NOBEL COATINGS INT BV 2014-08-13 CN disclosed
EP-2513237-B1 STAIN-BLOCKING AQUEOUS COATING COMPOSITION AKZO NOBEL COATINGS INT BV (NL) 2014-06-18 EP disclosed
WO-2011073164-A1 STAIN-BLOCKING AQUEOUS COATING COMPOSITION AKZO NOBEL COATINGS INTERNATIONAL B.V. (NL) 2011-06-23 WO disclosed
EP-0121192-B1 ANALYTICAL TEST COMPOSITION, DEVICE, METHOD FOR ITS PREPARATION AND METHOD FOR THE DETERMINATION OF PEROXIDATIVELY ACTIVE SUBSTANCE MILES INC. (US) 1990-06-27 EP disclosed
EP-0310061-A1 5-Mono or Disubstituted-3-(phenyl or 2-naphthalenyl)-3-[(1H-imidazol-1-ylmethyl) or (1H-1,2,4-triazol-1-ylmethyl)]-2-(methyl or benzyl)isoxazolidines FISONS CORPORATION (US) 1989-04-05 EP disclosed
US-4785117-A 5,5-disubstituted-3-phenyl-3-phenyl-3-[(1H-imidazol-1-ylmethyl) or (1H-1,2,4-triazol-1-ylmethyl)]-2-methylisoxazolidine derivatives (IR 3012) PENNWALT CORPORATION (US) 1988-11-15 US disclosed
US-4650910-A CLEAVAGE OF N-ACYL-B-PHENETHYLAMINES WITH BASE BAYER AKTIENGESELLSCHAFT (DE) 1987-03-17 US disclosed
EP-0197274-A1 Process for the preparation of substituted styrenes BAYER AG (DE) 1986-10-15 EP disclosed
EP-0121192-A2 Analytical test composition, device, method for its preparation and method for the determination of peroxidatively active substance MILES INC. (US) 1984-10-10 EP disclosed
US-4447542-A USING SUBSTITUTED CUMENE HYDROPEROXIDE AND INDICATOR; COLORIMETRIC ANALYSIS MILES LABORATORIES, INC. (US) 1984-05-08 US disclosed
US-4085165-A ISOCYANATE PREPOLYMER, VINYL COMPOUND, POLYAMINE OR POLYETHER CURING AGENT BRIDGESTONE TIRE CO., LTD. (JA) 1978-04-18 US disclosed
US-4016341-A REDUCING SCALE DEPOSITS BY COATING SURFACES WITH PHOSPHORIC ESTERS OR SALTS SHIN-ETSU CHEMICAL COMPANY LIMITED (JA) 1977-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240199558-A1 2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CX3CR1 CX3CR1, CCR2, CCR5 TSHR 1113/4885NPFFR2 848/4885SRD5A2 1896/4885
US-20240383866-A1 2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CX3CR1 CX3CR1, CCR2, CCR5 TSHR 1113/4885NPFFR2 848/4885SRD5A2 1896/4885
US-12404253-B2 2,4,6-trisubstituted 1,3,5-triazines as modulators of CX3CR1 CX3CR1, CCR2, CCR5 TSHR 1113/4885NPFFR2 848/4885SRD5A2 1896/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.