SCHEMBL2016173

SCHEMBL2016173

CCn1c(CNC(=O)c2nc(Cl)c(N)nc2N)nc2cc(S(C)(=O)=O)ccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.42
GAA P10253 2/20 0.42
S1PR1 P21453 2/20 0.40
HDAC6 Q9UBN7 1/20 0.39
RORC P51449 5/20 0.39
PPARG P37231 1/20 0.39
LMNA P02545 3/20 0.39
HPGD P15428 2/20 0.39
CYP1A2 P05177 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GMNN O75496 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
NFKB1 P19838 1/20 0.39
THPO P40225 1/20 0.39
STAT6 P42226 1/20 0.39
RECQL P46063 1/20 0.39
PMP22 Q01453 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2019895 0.86 HTT (0.44) HTTHDAC6PPARGLMNACYP1A2
Iodide SCHEMBL2019374 0.85 HTT (0.43) HTTHDAC6PPARGLMNACYP1A2
SCHEMBL2019532 0.85 HDAC6 (0.49) HTTGAAHDAC6PPARGHPGD
SCHEMBL2015349 0.83 HTT (0.57) HTTGAALMNAHPGDSMN1; SMN2
SCHEMBL2018490 0.83 KDM4E (0.53) HTTHDAC6KDM4EALDH1A1RECQL
SCHEMBL2014471 0.82 MAPT (0.52) HTTGAAHDAC6HPGDKDM4E
SCHEMBL2040435 0.82 HTT (0.45) HTTGAALMNACYP1A2SMN1; SMN2
SCHEMBL2014103 0.81 SCNN1A (0.43) HTTGAAHDAC6PPARGSMN1; SMN2
SCHEMBL2014823 0.81 HTT (0.45) HTTLMNACYP1A2CYP3A4CYP2D6
SCHEMBL2016331 0.81 HTT (0.52) HTTGAALMNAHPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed