SCHEMBL20145231

SCHEMBL20145231

Clc1ccc(NC2CCCN(Oc3ncccc3-c3ncccn3)C2)nc1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.43
HCRTR1 O43613 11/20 0.41
HCRTR2 O43614 4/20 0.39
CCNK O75909 1/20 0.38
CDK12 Q9NYV4 1/20 0.38
TSHR P16473 3/20 0.37
GAA P10253 2/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.35
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20144970 0.77 HCRTR1 (0.52) HCRTR1HCRTR2CCNKCDK12
SCHEMBL20144983 0.72 HCRTR1 (0.52) HCRTR1HCRTR2CCNKCDK12
SCHEMBL20145164 0.72 HCRTR1 (0.52) HCRTR1HCRTR2CCNKCDK12
SCHEMBL20145228 0.71 IL1B (0.54) CCNKCDK12
SCHEMBL20144912 0.70 HCRTR1 (0.56) HCRTR1HCRTR2CCNKCDK12
SCHEMBL20145167 0.69 CCNK (0.48) HCRTR1HCRTR2CCNKCDK12TSHR
SCHEMBL16147979 0.68 HCRTR1 (0.76) HCRTR1HCRTR2
SCHEMBL20145009 0.67 GFER (0.49) HCRTR1HCRTR2CCNKCDK12
SCHEMBL15739537 0.65 HCAR3 (0.56) PDE10ACCNKCDK12TSHRKDM4E
SCHEMBL16147928 0.64 HCRTR1 (0.68) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed