SCHEMBL2014551

SCHEMBL2014551

CC(C)(C)OC(=O)N1CCN(c2cccnc2-c2ccc3c(c2)C(C)(C)CCC3(C)C)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.46
POLB P06746 1/20 0.45
CKS1B P61024 2/20 0.45
SKP1 P63208 2/20 0.45
SKP2 Q13309 2/20 0.45
SMARCA2 P51531 1/20 0.43
SMARCA4 P51532 1/20 0.43
PBRM1 Q86U86 1/20 0.43
GPR119 Q8TDV5 4/20 0.42
KIT P10721 2/20 0.42
ACHE P22303 1/20 0.41
SQOR Q9Y6N5 1/20 0.41
RET P07949 1/20 0.40
DTYMK P23919 1/20 0.40
PDK2 Q15119 1/20 0.40
PIK3CA P42336 1/20 0.40
GBA1 P04062 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014735 0.82 WNT3A (0.46) CKS1BSKP1SKP2GPR119ACHE
SCHEMBL9961630 0.81 CKS1B (0.65) AKT1POLBCKS1BSKP1SKP2
SCHEMBL2015814 0.80 ACHE (0.52) CKS1BSKP1SKP2GPR119ACHE
SCHEMBL8514101 0.80 GPR119 (0.43) CKS1BSKP1SKP2SMARCA2SMARCA4
SCHEMBL3637662 0.80 GRIA1 (0.55) AKT1POLBCKS1BSKP1SKP2
SCHEMBL2017261 0.80 GPR119 (0.49) CKS1BSKP1SKP2GPR119PDK2
SCHEMBL2015195 0.80 CKS1B (0.46) CKS1BSKP1SKP2GPR119ACHE
SCHEMBL8515152 0.79 GPR119 (0.48) CKS1BSKP1SKP2GPR119KIT
SCHEMBL2015994 0.79 RARA (0.50) CKS1BSKP1SKP2SMARCA2SMARCA4
SCHEMBL12632947 0.79 RARG (0.48) SMARCA2SMARCA4PBRM1GPR119PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513057-A1 SPHINGOSINE KINASE INHIBITORS Merck Patent GmbH (DE) 2012-10-24 EP disclosed
WO-2011072791-A1 SPHINGOSINE KINASE INHIBITORS MERCK PATENT GMBH (DE) 2011-06-23 WO disclosed