SCHEMBL2015518

SCHEMBL2015518

C[Si](C)(C)C#Cc1c(F)cc(CC=O)c(-c2cccc(F)c2)c1N

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.32
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
TAAR1 Q96RJ0 2/20 0.31
PTPN11 Q06124 1/20 0.31
MTOR P42345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2013163 0.83 FBP1 (0.31)
SCHEMBL2015516 0.78 TRPM8 (0.36) ADORA1ADORA2AADORA2BTAAR1PTPN11
SCHEMBL2013731 0.72 AR (0.36) ADORA1ADORA2ATAAR1PTPN11
SCHEMBL3907818 0.69 AR (0.41) TAAR1
SCHEMBL2015127 0.67 CSNK1D (0.35) ADORA1
SCHEMBL2015218 0.67 CDC7 (0.40)
SCHEMBL7493782 0.65 TAAR1 (0.50) TAAR1
SCHEMBL14783969 0.65 DCLRE1B (0.47) TAAR1
SCHEMBL18097560 0.64 FFAR1 (0.34)
SCHEMBL2013162 0.64 FBP1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed