SCHEMBL20155378

SCHEMBL20155378

CCNSc1ccc(Oc2ccc(F)cc2F)c(B(O)O)c1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 7/20 0.35
CARM1 Q86X55 1/20 0.33
HSPB1 P04792 1/20 0.33
BRD4 O60885 6/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20154947 0.82 EPAS1 (0.45) TRPA1HSPB1BRD4
SCHEMBL28505143 0.73 ENPP2 (0.48) TRPA1HSPB1
SCHEMBL20155313 0.73 MEP1B (0.43) BRD4
SCHEMBL16651491 0.72 BRD4 (0.55) BRD4
SCHEMBL15068027 0.70 SCN8A (0.46) TRPA1BRD4
SCHEMBL10456772 0.67 TRPA1 (0.56) TRPA1HSPB1
SCHEMBL29952296 0.64 L3MBTL1 (0.42)
SCHEMBL1440694 0.64 L3MBTL1 (0.42)
SCHEMBL39406 0.64 CES2 (0.43)
SCHEMBL29395656 0.64 CES2 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed