SCHEMBL20157191

SCHEMBL20157191

C=C(Cl)/C=C(/Cl)CC(OC)N1CCN(c2ccccc2C#N)CC1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.40
DPP4 P27487 1/20 0.39
DRD2 P14416 7/20 0.39
DRD4 P21917 7/20 0.39
GRM5 P41594 1/20 0.39
DRD3 P35462 4/20 0.39
MC4R P32245 1/20 0.38
HTR7 P34969 4/20 0.38
HTR1A P08908 3/20 0.38
HSP90AB1 P08238 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
HTR2A P28223 1/20 0.37
THPO P40225 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157179 0.83 HSP90AB1 (0.39) THRBDPP4DRD2DRD4GRM5
SCHEMBL20157218 0.81 HTR7 (0.40) THRBDPP4DRD2DRD4DRD3
SCHEMBL20156862 0.71 DRD2 (0.45) THRBDRD2DRD4GRM5DRD3
SCHEMBL20156961 0.68 DRD2 (0.49) DRD2DRD4GRM5DRD3MC4R
SCHEMBL13898671 0.68 MC4R (0.51) DRD2DRD4GRM5DRD3MC4R
SCHEMBL3088832 0.67 DRD4 (0.54) DRD2DRD4GRM5DRD3HTR7
SCHEMBL14355275 0.65 HSP90AB1 (0.66) DRD2DRD3HTR7HTR1AHSP90AB1
SCHEMBL8760562 0.65 DRD2 (0.43) DPP4DRD2DRD4GRM5DRD3
SCHEMBL20156977 0.65 HTR7 (0.47) THRBDRD2DRD4GRM5DRD3
SCHEMBL9118895 0.63 DRD2 (0.45) THRBDRD2DRD4GRM5DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed