SCHEMBL20157472

SCHEMBL20157472

C=Cc1ccc(C(=O)c2ccc(CBr)cc2Br)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
LSS P48449 4/20 0.36
TAS1R3 Q7RTX0 2/20 0.34
TAS1R1 Q7RTX1 2/20 0.34
HPGD P15428 1/20 0.33
RXRA P19793 1/20 0.33
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TGM2 P21980 1/20 0.32
ALDH1A1 P00352 1/20 0.31
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
SRD5A2 P31213 2/20 0.31
AKR1C3 P42330 1/20 0.30
PTPN1 P18031 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362746 0.82 TAS1R3 (0.35) LSSTAS1R3TAS1R1HPGDRXRA
SCHEMBL20157960 0.81 SRD5A2 (0.49) CES2CES1RXRAMAPTHTT
SCHEMBL20157297 0.81 GSK3B (0.43) CES2CES1MAPTALDH1A1CYP4F2
SCHEMBL20157560 0.81 PTPN1 (0.43) CES2CES1MAPTHTTSMN1; SMN2
SCHEMBL21362533 0.78 ACHE (0.43) LSSHPGDMAPTALDH1A1PTPN1
SCHEMBL20158073 0.78 LMNA (0.46) CES2CES1MAPTHTTSMN1; SMN2
SCHEMBL20157412 0.77 NPC1 (0.54) CES2CES1HPGDMAPTHTT
SCHEMBL14593132 0.73 CES2 (0.38) CES2CES1HPGDMAPTALDH1A1
SCHEMBL21362630 0.73 HPGD (0.38) LSSTAS1R3TAS1R1HPGDRXRA
SCHEMBL1018494 0.71 PTPN1 (0.47) CES2CES1HPGDSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed