SCHEMBL20170713

SCHEMBL20170713

COc1ccc2c(c1OCc1ccccc1)C1CC(=O)CCC1CC2

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 11/20 0.41
AGTR1 P30556 2/20 0.41
KDM1A O60341 2/20 0.39
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
HTR1A P08908 3/20 0.39
DRD2 P14416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170653 0.75 GAA (0.42) PDE4APDE4BPDE4CPDE4D
SCHEMBL28006262 0.69 GLRA1 (0.42) AGTR2AGTR1KDM1AMAOAMAOB
SCHEMBL18458090 0.67 GAA (0.44) AGTR2AGTR1PDE4APDE4BPDE4C
SCHEMBL10073579 0.67 AGTR2 (0.49) AGTR2AGTR1PDE4APDE4BPDE4C
SCHEMBL9323521 0.65 ALDH1A1 (0.64) AGTR2AGTR1MAOAMAOBHTR1A
SCHEMBL13301272 0.65 HTR1A (0.34) HTR1ADRD2
SCHEMBL21300617 0.65 BCHE (0.67) HTR1A
SCHEMBL20852458 0.65 NQO2 (0.41) DRD2
SCHEMBL2742557 0.65 AGTR2 (0.45) AGTR2AGTR1MAOAMAOBPDE4B
SCHEMBL20170725 0.65 HTR1A (0.36) KDM1AMAOAMAOBHTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed