SCHEMBL2017066

SCHEMBL2017066

NCCc1cc(Cl)c2cnoc2c1-c1cccc(F)c1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 7/20 0.43
NT5E P21589 1/20 0.34
GRM5 P41594 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
CCNT1 O60563 1/20 0.32
CDK9 P50750 1/20 0.32
ACLY P53396 1/20 0.32
MAOB P27338 3/20 0.32
DPP4 P27487 1/20 0.32
HRH1 P35367 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012666 0.79 TAAR1 (0.47) TAAR1NT5EMAOB
SCHEMBL2015154 0.78 TAAR1 (0.41) TAAR1NT5ECCNT1CDK9DPP4
SCHEMBL2015779 0.75 PIK3CD (0.44) TAAR1L3MBTL1
SCHEMBL12491178 0.74 BCL2 (0.47) TAAR1NT5EDPP4
SCHEMBL9952729 0.68 PIK3CD (0.44) TAAR1
Trifluoroacetic Acid SCHEMBL2012078 0.68 BCL2 (0.41) TAAR1NT5E
SCHEMBL9953114 0.68 TAAR1 (0.38) TAAR1
SCHEMBL9953794 0.67 TAAR1 (0.40) TAAR1
SCHEMBL9953176 0.67 LMNA (0.39) TAAR1L3MBTL1
SCHEMBL9953509 0.67 ADORA1 (0.40) TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed