SCHEMBL20170726

SCHEMBL20170726

CC12c3c4ccc(O)c3OC1C(O)CCC2CC4

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 10/20 0.43
OPRD1 P41143 8/20 0.38
SIGMAR1 Q99720 2/20 0.38
OPRK1 P41145 6/20 0.38
LMNA P02545 2/20 0.36
CYP1A2 P05177 1/20 0.36
PKM P14618 1/20 0.36
THPO P40225 1/20 0.36
MRGPRX2 Q96LB1 2/20 0.36
SLC22A1 O15245 1/20 0.36
ADRA2A P08913 1/20 0.36
ARRB1 P49407 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22559865 0.67 OPRM1 (0.43) OPRM1OPRD1SIGMAR1OPRK1MRGPRX2
SCHEMBL14542485 0.67 OPRM1 (0.43) OPRM1OPRD1SIGMAR1OPRK1MRGPRX2
SCHEMBL20170754 0.65 OPRM1 (0.41) OPRM1OPRD1SIGMAR1OPRK1
SCHEMBL20170829 0.64 OPRD1 (0.46) OPRM1OPRD1SIGMAR1OPRK1
Dihydromorphine SCHEMBL19615483 0.63 OPRD1 (0.71) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL13380388 0.63 OPRD1 (0.71) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL19645038 0.63 OPRD1 (0.71) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL26346 0.63 OPRD1 (0.71) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL17025853 0.63 OPRD1 (0.71) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL19107002 0.63 OPRD1 (0.71) OPRM1OPRD1OPRK1MRGPRX2SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed