SCHEMBL20170756

SCHEMBL20170756

CCCCNC1C2CCC(=O)C[C@]23CC1(C)c1c(/C=C/C(=O)OC)cc(OC)c(O)c13

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.34
GAA P10253 1/20 0.33
ALOX5 P09917 1/20 0.31
BCHE P06276 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170851 0.89 GAA (0.34) GAA
SCHEMBL20170664 0.84 GAA (0.36) TRPV1GAA
SCHEMBL20170619 0.78 TRPV1 (0.33) TRPV1ALOX5BCHE
SCHEMBL20170594 0.77 OPRM1 (0.33) TRPV1
SCHEMBL20170874 0.75 ALOX5 (0.33) GAAALOX5
SCHEMBL20170666 0.73 GAA (0.37) GAA
SCHEMBL21202074 0.73 GAA (0.47) TRPV1GAA
SCHEMBL20170821 0.71 GAA (0.36) GAA
SCHEMBL20170595 0.71 GAA (0.36) GAA
SCHEMBL12646160 0.68 OPRM1 (0.48) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed