SCHEMBL20170666

SCHEMBL20170666

C=CCNC1C2CCC(=O)C[C@]23CC1(C)c1c(Br)cc(OC)c(O)c13

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.37
HTR1A P08908 6/20 0.35
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32
HPGD P15428 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NR3C1 P04150 4/20 0.32
PGR P06401 2/20 0.32
AR P10275 2/20 0.32
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
IGF1R P08069 1/20 0.30
MEN1 O00255 1/20 0.30
HTT P42858 1/20 0.30
GFER P55789 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170821 0.87 GAA (0.36) GAAOPRM1
SCHEMBL20170664 0.87 GAA (0.36) GAASMN1; SMN2MEN1KMT2A
SCHEMBL20170718 0.81 GAA (0.36) GAAALDH1A1MAPTHPGDSMN1; SMN2
SCHEMBL20170595 0.77 GAA (0.36) GAA
SCHEMBL20170609 0.76 NR3C1 (0.33) GAANR3C1PGRAR
SCHEMBL10222587 0.75 GAA (0.39) GAAHTR1AALDH1A1MAPTHPGD
SCHEMBL20170707 0.75 GAA (0.35) GAAALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL20170874 0.75 ALOX5 (0.33) GAANR3C1PGRARMEN1
SCHEMBL20170851 0.75 GAA (0.34) GAA
SCHEMBL20170756 0.73 TRPV1 (0.34) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed