SCHEMBL20177642

SCHEMBL20177642

COc1ccc(COC(=O)N[C@@H]2c3nc4ccccc4n3C[C@H]2c2ccc(Br)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.39
PKM P14618 1/20 0.39
HTT P42858 1/20 0.39
GSK3B P49841 1/20 0.39
ALDH1A1 P00352 3/20 0.38
KMT2A Q03164 1/20 0.38
CNR2 P34972 3/20 0.38
MAPT P10636 1/20 0.38
KDM4E B2RXH2 2/20 0.37
NPC1 O15118 1/20 0.37
ATM Q13315 1/20 0.37
KCNH2 Q12809 1/20 0.36
KDM1A O60341 1/20 0.36
BRD4 O60885 1/20 0.36
BRD2 P25440 1/20 0.36
BRD3 Q15059 1/20 0.36
GRM2 Q14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177499 0.88 SMN1; SMN2 (0.37) SMN1; SMN2PKMHTTGSK3BALDH1A1
SCHEMBL20177659 0.81 HTT (0.40) SMN1; SMN2PKMHTTALDH1A1KMT2A
SCHEMBL20177557 0.80 CA1 (0.42) NPC1BRD4BRD2BRD3
SCHEMBL20177846 0.75 KDM1A (0.40) SMN1; SMN2PKMHTTALDH1A1KMT2A
SCHEMBL20177565 0.73 FPR1 (0.43) SMN1; SMN2PKMHTTALDH1A1KMT2A
SCHEMBL20177842 0.72 FPR1 (0.53)
SCHEMBL20177637 0.72 FPR1 (0.44) SMN1; SMN2PKMHTTALDH1A1KMT2A
SCHEMBL20177777 0.71 FPR2 (0.44) HTTALDH1A1KMT2AMAPTNPC1
SCHEMBL20177614 0.67 CTSL (0.42) ALDH1A1KMT2AKDM1A
SCHEMBL20177925 0.67 FPR2 (0.46) SMN1; SMN2PKMHTTALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed