SCHEMBL201886

SCHEMBL201886

CCCc1ccc(-c2ccccc2C(=O)N2C[C@H](O)[C@H](O)[C@H]2C(=O)NOCc2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MLNR O43193 1/20 0.37
CYP3A4 P08684 1/20 0.37
LMNA P02545 1/20 0.35
CHRNB2 P17787 4/20 0.35
CHRNA4 P43681 4/20 0.35
CHRNB4 P30926 3/20 0.35
CHRNA3 P32297 3/20 0.35
PPARG P37231 2/20 0.35
LTB4R2 Q9NPC1 2/20 0.35
KDM2B Q8NHM5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2693933 0.88 MMP13 (0.41)
SCHEMBL200909 0.88 CHRNB2 (0.38) MLNRCYP3A4LMNACHRNB2CHRNA4
SCHEMBL202876 0.86 MMP13 (0.43) MLNRCYP3A4PPARGKDM2B
SCHEMBL201196 0.83 LMNA (0.37) MLNRCYP3A4LMNACHRNB2CHRNA4
SCHEMBL201123 0.80 LMNA (0.37) MLNRCYP3A4LMNAPPARGLTB4R2
SCHEMBL203379 0.79 MMP13 (0.38) MLNRCYP3A4PPARGKDM2B
SCHEMBL201676 0.79 MMP13 (0.38) MLNRCYP3A4PPARGKDM2B
SCHEMBL200777 0.77 NPC1 (0.44)
SCHEMBL13530903 0.75 FFAR2 (0.36)
SCHEMBL10208064 0.75 FFAR2 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088804-B2 N-hydroxyamide derivatives possessing antibacterial activity PFIZER INC. (US) 2012-01-03 US disclosed
EP-2338878-A2 N-hydroxyamide derivatives possessing antibacterial activity Vicuron Pharmaceuticals, Inc. (US) 2011-06-29 EP disclosed
US-20100022605-A1 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY VICURON PHARMACEUTICALS INC. 2010-01-28 US disclosed
EP-1963262-A2 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY Vicuron Pharmaceuticals, Inc. (US) 2008-09-03 EP disclosed
WO-2007069020-A2 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY VICURON PHARMACEUTICALS INC. (US) 2007-06-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100022605-A1 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY NAAA, HDHD5, HACL2 MLNR 1501/4885CYP3A4 1791/4885LMNA 1020/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.