SCHEMBL20193251

SCHEMBL20193251

CS(C)(C)CCOCn1cc(-c2cn(S(=O)(=O)Cc3ccccc3)c3cnc(Br)cc23)cn1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 12/20 0.33
DYRK1B Q9Y463 1/20 0.33
BRD4 O60885 1/20 0.30
ALK Q9UM73 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16608489 0.90 DGAT1 (0.35) CREBBPDYRK1BBRD4ALK
SCHEMBL20193242 0.86 CHUK (0.36)
SCHEMBL20193181 0.86 CHUK (0.40) CREBBPDYRK1BALK
SCHEMBL20193252 0.85 HTR6 (0.33)
SCHEMBL20193264 0.84 CHUK (0.49)
SCHEMBL20193178 0.82 L3MBTL1 (0.39) BRD4ALK
SCHEMBL20193179 0.81 CREBBP (0.32) CREBBPBRD4ALKCYP2C19
SCHEMBL19114543 0.80 CHUK (0.35) CREBBP
SCHEMBL20193151 0.78 CHUK (0.34)
SCHEMBL20193217 0.78 DYRK1A (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9981963-B2 3-(1H-pyrazol-4-yl)-1H-pyrrolo[2,3-c]pyridine derivatives as NIK inhibitors JANSSEN PHARMACEUTICA NV (BE) 2018-05-29 US disclosed