SCHEMBL20195459

SCHEMBL20195459

CN(N)C(=O)N(N)c1cccc(F)c1COc1ccccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.38
GABRA5 P31644 2/20 0.36
TSHR P16473 1/20 0.36
GRM5 P41594 4/20 0.35
TDP1 Q9NUW8 2/20 0.34
ALDH1A1 P00352 2/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HCRTR2 O43614 2/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GUCY1B2 O75343 2/20 0.32
GUCY1A2 P33402 2/20 0.32
GUCY1A1 Q02108 2/20 0.32
GUCY1B1 Q02153 2/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
HCRTR1 O43613 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20195402 0.87 GABRA5 (0.39) GABRA5TSHRGRM5ALDH1A1L3MBTL1
SCHEMBL20195398 0.84 RXFP1 (0.36) ADORA2AGABRA5GRM5ALDH1A1KMT2A
SCHEMBL20195455 0.84 NPC1 (0.38) GABRA5TSHRGRM5ALDH1A1NPC1
SCHEMBL22037265 0.84 FFAR4 (0.35) GABRA5KMT2ARAB9ASMN1; SMN2
SCHEMBL20195604 0.84 GABRA5 (0.38) GABRA5ALDH1A1HCRTR2HCRTR1
SCHEMBL20845040 0.81 SLC16A3 (0.32) TDP1ALDH1A1KMT2AATML3MBTL1
SCHEMBL20195410 0.78 SGMS2 (0.42) TSHRTDP1ALDH1A1KMT2AATM
SCHEMBL18831653 0.77 MRGPRX4 (0.40) GRM5RAB9AGUCY1B2GUCY1A2GUCY1A1
SCHEMBL16446199 0.75 GABRA5 (0.47) ADORA2AGABRA5GRM5ALDH1A1NPC1
SCHEMBL22590911 0.75 ALDH1A1 (0.33) TDP1ALDH1A1KMT2AL3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3029035-B1 TETRAZOLINONE COMPOUND, AND USE THEREOF SUMITOMO CHEMICAL CO (JP) 2018-05-30 EP disclosed