SCHEMBL20195612

SCHEMBL20195612

CCOc1cccc(OC#N)c1COc1nc(C)ccc1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 8/20 0.36
KDM4E B2RXH2 2/20 0.36
HSD17B10 Q99714 2/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
BDKRB2 P30411 1/20 0.34
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HPGD P15428 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20195639 0.85 BDKRB2 (0.42) SMN1; SMN2BDKRB2MAPTCYP1A2CYP3A4
SCHEMBL20195536 0.81 HTR6 (0.35) HSD17B10LMNABDKRB2TSHRCYP1A2
SCHEMBL20195589 0.81 ALDH1A1 (0.44) GRM5KDM4EHSD17B10NPC1LMNA
SCHEMBL20195628 0.77 TP53 (0.44) KDM4EHSD17B10NPC1LMNARAB9A
SCHEMBL18831616 0.77 ESR1 (0.38) KDM4EHSD17B10MAPTHTTHPGD
SCHEMBL20195606 0.73 GABRA5 (0.40) GRM5KDM4ENPC1SMN1; SMN2BDKRB2
SCHEMBL20195516 0.72 SYK (0.37) GRM5KDM4ENPC1LMNARAB9A
SCHEMBL17707924 0.72 GRM5 (0.42) GRM5KDM4EHSD17B10NPC1LMNA
SCHEMBL20195542 0.71 GABRA5 (0.43) GRM5NPC1RAB9ABDKRB2CYP1A2
SCHEMBL18831604 0.71 MAPT (0.40) KDM4ENPC1LMNARAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3029035-B1 TETRAZOLINONE COMPOUND, AND USE THEREOF SUMITOMO CHEMICAL CO (JP) 2018-05-30 EP disclosed