SCHEMBL2019650

SCHEMBL2019650

NC(=O)c1cccc(N)c1O

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.69
ALDH1A1 P00352 3/20 0.52
KDM4E B2RXH2 2/20 0.52
MAPT P10636 2/20 0.52
HSD17B10 Q99714 2/20 0.52
HPGD P15428 1/20 0.52
TSHR P16473 1/20 0.52
METAP2 P50579 1/20 0.43
CXCR2 P25025 1/20 0.42
GAA P10253 2/20 0.42
G6PD P11413 1/20 0.42
CASP7 P55210 1/20 0.42
CASP6 P55212 1/20 0.42
BCAT2 O15382 1/20 0.42
PARP1 P09874 3/20 0.41
IKBKB O14920 2/20 0.41
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
PDPK1 O15530 1/20 0.41
CFTR P13569 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL2026072 0.94 MMP2 (0.68) MMP2ALDH1A1KDM4EMAPTHSD17B10
Cadaverine Tartrate SCHEMBL2021423 0.87 MMP2 (0.59) MMP2ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL698742 0.85 KDM4E (0.61) MMP2ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL720049 0.84 MMP2 (0.72) MMP2ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL3723645 0.83 KDM4E (0.58) MMP2ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL29547161 0.82 MMP2 (1.00) MMP2ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL204392 0.82 MMP2 (1.00) MMP2ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL3378787 0.80 MMP2 (0.67) MMP2ALDH1A1KDM4EMAPTHSD17B10
Hydrochloric Acid SCHEMBL5110306 0.80 MMP2 (0.96) MMP2ALDH1A1KDM4EMAPTHSD17B10
Ammonia Solution, Strong SCHEMBL1224587 0.80 MMP2 (0.96) MMP2ALDH1A1KDM4EMAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 147 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8519168-B2 Process and intermediates for the synthesis of 1,2-substituted 3,4-dioxo-1-cyclobutene compounds MERCK SHARP & DOHME CORP. (US) 2013-08-27 US claimed
US-20110160469-A1 PROCESS AND INTERMEDIATES FOR THE SYNTHESIS OF 1,2-SUBSTITUTED 3,4-DIOXO-1-CYCLOBUTENE COMPOUNDS MERCK SHARP & DOHME LLC 2011-06-30 US claimed
CN-101932553-A Process and intermediates for the synthesis of 1,2-substituted 3,4-dioxo-1-cyclobutene compounds SCHERING CORP 2010-12-29 CN claimed
EP-2178826-A1 PROCESS AND INTERMEDIATES FOR THE SYNTHESIS OF 1,2-SUBSTITUTED 3,4-DIOXO-1-CYCLOBUTENE COMPOUNDS SCHERING CORPORATION (US) 2010-04-28 EP claimed
WO-2009005801-A1 PROCESS AND INTERMEDIATES FOR THE SYNTHESIS OF 1,2-SUBSTITUTED 3,4-DIOXO-1-CYCLOBUTENE COMPOUNDS SCHERING CORPORATION (US) 2009-01-08 WO claimed
EP-0970057-B1 SUBSTITUTED AMINOSALICYCLIC ACID AMIDES WITH FUNGICIDAL EFFECT AND INTERMEDIATE PRODUCTS FOR PRODUCTION THEREOF BAYER CROPSCIENCE AG (DE) 2006-02-01 EP claimed
CN-1121393-C Substituted aminosalicylamides having fungicidal action and intermediates for their preparation BAYER AG (DE) 2003-09-17 CN claimed
EP-0848700-B1 ACYLAMINOSALICYLIC ACID AMIDES AND THEIR USES AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2003-07-02 EP claimed
US-20020006958-A1 Substituted aminosalicylic acid amides with fungicidal effect and intermediate products for production thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2002-01-17 US claimed
US-6333432-B1 CONTROLLING PHYTOPATHOGENS DOW AGROSCIENCES LLC 2001-12-25 US claimed
EP-1035772-A4 FUNGICIDAL COMPOSITIONS AND METHODS, AND COMPOUNDS AND METHODS FOR THE PREPARATION THEREOF DOW AGROSCIENCES LLC (US) 2001-03-28 EP claimed
US-6194418-B1 Substituted aminosalicyclic acid amides with fungicidal effect and intermediate products for production thereof BAYER AKTIENGESELLSCHAFT (DE) 2001-02-27 US claimed
EP-1035772-A1 FUNGICIDAL COMPOSITIONS AND METHODS, AND COMPOUNDS AND METHODS FOR THE PREPARATION THEREOF Dow AgroSciences LLC (US) 2000-09-20 EP claimed
CN-1250442-A Substituted aminosalicylamides having fungicidal action and intermediates for their preparation BAYER AG (DE) 2000-04-12 CN claimed
US-6001879-A SUITABLE FOR CONTROLLING PESTS, PREFERABLY FUNGI, INSECTS AND BACTERIA, IN PLANTS AND INDUSTRIAL MATERIALS; METHODS OF THEIR SYBNTHESIS INCLUDING REACTING AMINOSALICYLAMIDES WITH ACYLATING AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1999-12-14 US claimed
WO-1999027783-A1 FUNGICIDAL COMPOSITIONS AND METHODS, AND COMPOUNDS AND METHODS FOR THE PREPARATION THEREOF DOW AGROSCIENCES LLC (US) 1999-06-10 WO claimed
US-12454507-B2 Compounds having a fungicidal activity, their agronomic compositions and use thereof for the control of phytopathogenic fungi ISAGRO SPA (IT) 2025-10-28 US disclosed
US-20240116855-A1 COMPOUNDS HAVING A FUNGICIDAL ACTIVITY, THEIR AGRONOMIC COMPOSITIONS AND USE THEREOF FOR THE CONTROL OF PHYTOPATHOGENIC FUNGI ISAGRO S.P.A. (IT) 2024-04-11 US disclosed
US-5648470-A Phenylboronic acid complexing reagents derived from aminosalicyclic acid PROLINX, INC. (US) 1997-07-15 US disclosed
US-5382502-A Photography, simplified synthesis EASTMAN KODAK COMPANY (US) 1995-01-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240116855-A1 COMPOUNDS HAVING A FUNGICIDAL ACTIVITY, THEIR AGRONOMIC COMPOSITIONS AND USE THEREOF FOR THE CONTROL OF PHYTOPATHOGENIC FUNGI CYP51A1, ERG28, DPM1 MMP2 724/4885ALDH1A1 771/4885KDM4E 1149/4885
US-20110160469-A1 PROCESS AND INTERMEDIATES FOR THE SYNTHESIS OF 1,2-SUBSTITUTED 3,4-DIOXO-1-CYCLOBUTENE COMPOUNDS CCL2, CCR1, CXCR1 MMP2 2261/4885ALDH1A1 1721/4885KDM4E 4463/4885
US-20020006958-A1 Substituted aminosalicylic acid amides with fungicidal effect and intermediate products for production thereof AADAC, DDC, DAO MMP2 1072/4885ALDH1A1 353/4885KDM4E 1414/4885
US-12454507-B2 Compounds having a fungicidal activity, their agronomic compositions and use thereof for the control of phytopathogenic fungi CYP51A1, ERG28, DPM1 MMP2 724/4885ALDH1A1 771/4885KDM4E 1149/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.