SCHEMBL2024281

SCHEMBL2024281

Cc1cc(O[Si](C)(C)C(C)(C)C)cc(C)c1-c1cccc(C=O)n1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.36
CA1 P00915 4/20 0.36
CA9 Q16790 4/20 0.36
PREP P48147 1/20 0.33
TERT O14746 3/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12578156 0.78 ALDH1A1 (0.44) CA12CA1CA9
SCHEMBL25391492 0.77 TERT (0.41) TERT
SCHEMBL30570368 0.77 TERT (0.41) TERT
SCHEMBL12577789 0.77 CA12 (0.34) CA12CA1CA9PREP
SCHEMBL3340077 0.75 HTR7 (0.41) TERT
SCHEMBL2027100 0.75 BRD4 (0.49) CA12CA1CA9PREPHSP90AA1
SCHEMBL12640965 0.75 TERT (0.40) TERTHSP90AA1
SCHEMBL13117421 0.74 PREP (0.35) CA12CA1CA9PREPHSP90AA1
SCHEMBL5799300 0.73 CA12 (0.37) CA12CA1CA9PREPTERT
SCHEMBL1251338 0.73 CA12 (0.40) CA12CA1CA9PREPHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7968552-B2 Oxadiazolidinedione compound ASTELLAS PHARMA INC. (JP) 2011-06-28 US disclosed
US-7968552-B2 Oxadiazolidinedione compound ASTELLAS PHARMA INC. (JP) 2011-06-28 US disclosed
US-20090186909-A1 Oxadiazolidinedione Compound ASTELLAS PHARMA INC. (JP) 2009-07-23 US disclosed
US-20090186909-A1 Oxadiazolidinedione Compound ASTELLAS PHARMA INC. (JP) 2009-07-23 US disclosed
EP-2011788-A1 OXADIAZOLIDINEDIONE COMPOUND Astellas Pharma Inc. (JP) 2009-01-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090186909-A1 Oxadiazolidinedione Compound GPR119, GPR39, GPR65 CA12 4396/4885CA1 4091/4885CA9 3645/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.