SCHEMBL20299385

SCHEMBL20299385

CC(=O)SCOC(=O)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.38
POLB P06746 2/20 0.33
GAA P10253 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TKT P29401 1/20 0.33
BTN3A1 O00481 4/20 0.33
CYP2C19 P33261 1/20 0.32
BLM P54132 1/20 0.31
ATM Q13315 1/20 0.31
ELANE P08246 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7348874 0.82 PRKCA (0.38) PRKCAPOLBGAANPSR1TKT
SCHEMBL6991459 0.78 PRKCA (0.42) PRKCAPOLBGAANPSR1BTN3A1
SCHEMBL12360855 0.76 PRKCA (0.41) PRKCAPOLBGAANPSR1BTN3A1
SCHEMBL6991468 0.74 PRKCA (0.39) PRKCAPOLBGAANPSR1BTN3A1
SCHEMBL14681224 0.71
SCHEMBL15837494 0.71 CYP2C19 (0.34) POLBGAACYP2C19BLMATM
SCHEMBL7348875 0.71 PRKCA (0.37) PRKCAPOLBGAANPSR1TKT
SCHEMBL767191 0.70 NAAA (0.40) POLBGAACYP2C19BLMATM
SCHEMBL14675199 0.70 CYP2C19 (0.33) POLBCYP2C19BLMATM
SCHEMBL681950 0.69 PRKCA (0.46) PRKCAPOLBGAANPSR1BTN3A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11001577-B2 Pesticidally active azetidine sulfones amide isoxazoline derivatives SYNGENTA PARTICIPATIONS AG (CH) 2021-05-11 US disclosed
US-11001577-B2 Pesticidally active azetidine sulfones amide isoxazoline derivatives SYNGENTA PARTICIPATIONS AG (CH) 2021-05-11 US disclosed
EP-3555083-B1 PESTICIDALLY ACTIVE AZETIDINE SULFONES AMIDE ISOXAZOLINE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2021-01-20 EP disclosed
EP-3555083-B1 PESTICIDALLY ACTIVE AZETIDINE SULFONES AMIDE ISOXAZOLINE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2021-01-20 EP disclosed
US-20200123143-A1 PESTICIDALLY ACTIVE AZETIDINE SULFONES AMIDE ISOXAZOLINE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2020-04-23 US disclosed
US-20200123143-A1 PESTICIDALLY ACTIVE AZETIDINE SULFONES AMIDE ISOXAZOLINE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2020-04-23 US disclosed
EP-3555083-A1 PESTICIDALLY ACTIVE AZETIDINE SULFONES AMIDE ISOXAZOLINE DERIVATIVES Syngenta Participations AG (CH) 2019-10-23 EP disclosed
WO-2018114791-A1 PESTICIDALLY ACTIVE AZETIDINE SULFONES AMIDE ISOXAZOLINE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2018-06-28 WO disclosed
WO-2018114791-A1 PESTICIDALLY ACTIVE AZETIDINE SULFONES AMIDE ISOXAZOLINE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2018-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200123143-A1 PESTICIDALLY ACTIVE AZETIDINE SULFONES AMIDE ISOXAZOLINE DERIVATIVES ACHE, PRDX1, DDT PRKCA 2753/4885POLB 4117/4885GAA 2076/4885
US-11001577-B2 Pesticidally active azetidine sulfones amide isoxazoline derivatives ACHE, PRDX1, DDT PRKCA 2753/4885POLB 4117/4885GAA 2076/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.