SCHEMBL2030928

SCHEMBL2030928

N#C/C=C/c1c(F)cccc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 4/20 0.35
SLC22A12 Q96S37 5/20 0.33
AR P10275 3/20 0.33
PTGES2 Q9H7Z7 1/20 0.33
PGR P06401 1/20 0.33
KIF11 P52732 1/20 0.33
ENPP2 Q13822 1/20 0.33
HSD11B1 P28845 1/20 0.31
NFKB1 P19838 1/20 0.31
KCNH2 Q12809 2/20 0.30
MAT2A P31153 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2030929 1.00 NFE2L2 (0.35) NFE2L2SLC22A12ARPTGES2PGR
SCHEMBL18215497 0.77 NFE2L2 (0.38) NFE2L2SLC22A12PTGES2HSD11B1NFKB1
SCHEMBL12641533 0.77 NFE2L2 (0.38) NFE2L2SLC22A12PTGES2HSD11B1NFKB1
SCHEMBL7484296 0.75 KCNH2 (0.47) KCNH2MAT2A
SCHEMBL7484292 0.75 KCNH2 (0.47) KCNH2MAT2A
SCHEMBL5644762 0.73 NFKB1 (0.53) NFKB1
SCHEMBL4728560 0.73 NFKB1 (0.53) NFKB1
SCHEMBL18215568 0.72 NFE2L2 (0.35) NFE2L2SLC22A12PTGES2HSD11B1KCNH2
SCHEMBL9683791 0.72 NFKB1 (0.38) ARENPP2HSD11B1NFKB1
SCHEMBL20086556 0.72 P2RX7 (0.37) NFE2L2SLC22A12ARPTGES2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012175514-A1 PYRIDINONE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-12-27 WO disclosed
WO-2011076687-A1 PYRIDINONE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-06-30 WO disclosed