SCHEMBL2033387

SCHEMBL2033387

CCOC(=O)C(=CC(C)CCC1=C(C)CCCC1(C)C)C(=O)OCC

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 5/20 0.43
RARB P10826 2/20 0.39
RARG P13631 2/20 0.39
RXRA P19793 2/20 0.39
RARA P10276 1/20 0.39
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 1/20 0.35
ACE2 Q9BYF1 2/20 0.35
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
ALOX5 P09917 1/20 0.34
ALOX15 P16050 1/20 0.34
GLO1 Q04760 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1636049 0.89 TRPA1 (0.46) TRPA1RARBRARGRXRARARA
SCHEMBL18084307 0.88 TRPA1 (0.41) TRPA1RARBRARGRXRARARA
SCHEMBL9205463 0.85 TRPA1 (0.40) TRPA1RARBRARGRXRARARA
SCHEMBL2039596 0.85 RARB (0.45) TRPA1RARBRARGRXRARARA
SCHEMBL9953603 0.84 TRPA1 (0.44) TRPA1RARBRARGRXRARARA
SCHEMBL16606707 0.84 TRPA1 (0.44) TRPA1RARBRARGRXRARARA
SCHEMBL10044179 0.84 TRPA1 (0.44) TRPA1RARBRARGRXRARARA
SCHEMBL18084338 0.81 TRPA1 (0.43) TRPA1RARBRARGRXRARARA
SCHEMBL13554953 0.79 ALDH1A1 (0.41) TRPA1RARBRARGRXRARARA
SCHEMBL9202801 0.77 TRPA1 (0.42) TRPA1RARBRARGRXRARARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3268346-B1 PROCESSES FOR THE PREPARATION OF UNSATURATED MALONATES INT FLAVORS & FRAGRANCES INC (US) 2021-05-05 EP disclosed
US-10358415-B2 Processes for the preparation of unsaturated malonates INTERNATIONAL FLAVORS & FRAGRANCES INC. (US) 2019-07-23 US disclosed
EP-2513030-B2 BETA-GAMMA UNSATURATED ESTERS AND PROCESS OF PRODUCTION OF BETA-GAMMA UNSATURATED ESTERS. GIVAUDAN SA (CH) 2018-08-29 EP disclosed
US-20180105490-A1 PROCESSES FOR THE PREPARATION OF UNSATURATED MALONATES INTERNATIONAL FLAVORS AND FRAGRANCES INC. 2018-04-19 US disclosed
US-20180105490-A1 PROCESSES FOR THE PREPARATION OF UNSATURATED MALONATES INTERNATIONAL FLAVORS AND FRAGRANCES INC. 2018-04-19 US disclosed
WO-2016145288-A1 PROCESSES FOR THE PREPARATION OF UNSATURATED MALONATES INTERNATIONAL FLAVORS & FRAGRANCES INC. (US) 2016-09-15 WO disclosed
EP-2513030-B1 BETA-GAMMA UNSATURATED ESTERS AND PROCESS OF PRODUCTION OF BETA-GAMMA UNSATURATED ESTERS. GIVAUDAN SA (CH) 2015-05-06 EP disclosed
US-8765980-B2 Organic compounds GIVAUDAN S.A. (CH) 2014-07-01 US disclosed
US-8765980-B2 Organic compounds GIVAUDAN S.A. (CH) 2014-07-01 US disclosed
US-8765980-B2 Organic compounds GIVAUDAN S.A. (CH) 2014-07-01 US disclosed
US-20120271059-A1 Organic Compounds GIVAUDAN SA (CH) 2012-10-25 US disclosed
US-20120271059-A1 Organic Compounds GIVAUDAN SA (CH) 2012-10-25 US disclosed
US-20120271059-A1 Organic Compounds GIVAUDAN SA (CH) 2012-10-25 US disclosed
EP-2513030-A1 ORGANIC COMPOUNDS Givaudan SA (CH) 2012-10-24 EP disclosed
WO-2011073387-A1 ORGANIC COMPOUNDS GIVAUDAN SA (CH) 2011-06-23 WO disclosed
WO-2011073387-A1 ORGANIC COMPOUNDS GIVAUDAN SA (CH) 2011-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10358415-B2 Processes for the preparation of unsaturated malonates ME1, ACSL6, MAL2 TRPA1 4202/4885RARB 87/4885RARG 92/4885
US-20120271059-A1 Organic Compounds HSD17B12, HSD17B1, MAL2 TRPA1 2304/4885RARB 408/4885RARG 568/4885
US-20180105490-A1 PROCESSES FOR THE PREPARATION OF UNSATURATED MALONATES ME1, ACSL6, MAL2 TRPA1 4202/4885RARB 87/4885RARG 92/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.