SCHEMBL20339367

SCHEMBL20339367

O=Cc1ccnc(-c2ccc(C(=O)O)cc2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
KMT2A Q03164 2/20 0.54
MPI P34949 1/20 0.54
LOXL2 Q9Y4K0 1/20 0.44
KDM4E B2RXH2 4/20 0.42
ERN1 O75460 2/20 0.41
TRIM24 O15164 1/20 0.41
TRIM33 Q9UPN9 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CAMK2D Q13557 2/20 0.41
MAP4K4 O95819 1/20 0.41
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40
BCL2L1 Q07817 1/20 0.39
BAD Q92934 1/20 0.39
MEN1 O00255 1/20 0.39
PRNP P04156 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18002781 0.82 KMT2A (0.52) ALDH1A1KMT2AMPIKDM4EMEN1
SCHEMBL12538607 0.79 KMT2A (0.51) ALDH1A1KMT2AMPIKDM4ETDP1
SCHEMBL2678442 0.79 ALDH1A1 (0.49) ALDH1A1KMT2AMPIERN1TSHR
SCHEMBL4585500 0.78 CCR1 (0.46) ALDH1A1KMT2AMPITRIM24TRIM33
SCHEMBL20339991 0.77 ERN1 (0.53) ALDH1A1LOXL2KDM4EERN1TRIM24
SCHEMBL20339735 0.76 RXRA (0.46) ALDH1A1KMT2ALOXL2KDM4ECAMK2D
SCHEMBL22320609 0.75 KMT2A (0.47) ALDH1A1KMT2AMPIKDM4EMAP4K4
SCHEMBL12151205 0.75 ALDH1A1 (0.47) ALDH1A1KMT2AMPI
SCHEMBL4899395 0.75 CAMK2D (0.64) KMT2AKDM4ECAMK2DMAP4K4MEN1
SCHEMBL1222172 0.74 MKNK1 (0.55) ALDH1A1KDM4EMKNK1MKNK2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200123146-A1 HETEROCYCLIC INTEGRIN AGONISTS GB006 INC (US) 2020-04-23 US disclosed
US-20200123146-A1 HETEROCYCLIC INTEGRIN AGONISTS GB006 INC (US) 2020-04-23 US disclosed
WO-2018126072-A1 HETEROCYCLIC INTEGRIN AGONISTS ADHAERE PHARMACEUTICALS, INC. (US) 2018-07-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200123146-A1 HETEROCYCLIC INTEGRIN AGONISTS ITGA1, ITGA4, ITGA2 ALDH1A1 1447/4885KMT2A 2000/4885MPI 2461/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.