SCHEMBL20401410

SCHEMBL20401410

O=C(O)c1cc(F)c(NCc2ccc(C3CCCCC3)cc2)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 3/20 0.46
HAO1 Q9UJM8 1/20 0.45
KMO O15229 1/20 0.45
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
KDM4C Q9H3R0 1/20 0.44
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
KMT2A Q03164 1/20 0.42
PPARA Q07869 1/20 0.41
VNN1 O95497 1/20 0.41
ACMSD Q8TDX5 1/20 0.41
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
SSTR3 P32745 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20400797 0.85 KDM4C (0.50) STAT3HAO1KMOHTR2CHTR2B
SCHEMBL20401012 0.85 S1PR1 (0.46) STAT3HAO1KMOHTR2CHTR2B
SCHEMBL20401408 0.84 STAT3 (0.49) STAT3MEN1ALDH1A1KMT2A
SCHEMBL2647028 0.79 HAO1 (0.52) HAO1KMOHTR2CHTR2BKDM4C
SCHEMBL20400984 0.76 S1PR1 (0.49) STAT3HAO1KMOHTR2CHTR2B
SCHEMBL20401001 0.76 SERPINE1 (0.51) STAT3HAO1KMOHTR2CHTR2B
SCHEMBL2377234 0.74 VNN1 (0.55) ALDH1A1POLBPPARAVNN1
SCHEMBL20401023 0.73 ALOX15 (0.53) STAT3KDM4CMEN1ALDH1A1KMT2A
SCHEMBL17084777 0.72 ACMSD (0.52) STAT3HTR2CHTR2BKDM4CPPARA
SCHEMBL354930 0.71 KMO (0.62) HAO1KMOMEN1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018136935-A1 2-ARYLSULFONAMIDO-N-ARYLACETAMIDE DERIVATIZED STAT3 INHIBITORS UNIVERSITY OF HAWAII (US) 2018-07-26 WO disclosed