Oxyquinoline

Oxyquinoline

SCHEMBL2042993

O=P(O)(O)O.Oc1cccc2cccnc12

nearest known ligand 0.81

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Oxyquinoline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A known ✓ P35348 1/20 0.81
KDR known ✓ P35968 1/20 0.45
TSHR P16473 3/20 0.81
MMP2 P08253 2/20 0.81
CHRM1 P11229 1/20 0.81
COMT P21964 1/20 0.81
METAP2 P50579 1/20 0.81
METAP1 P53582 1/20 0.81
HDAC8 Q9BY41 1/20 0.81
KDM4E B2RXH2 8/20 0.73
ALOX12 P18054 3/20 0.73
LMNA P02545 3/20 0.63
ALDH1A1 P00352 3/20 0.63
TDP1 Q9NUW8 4/20 0.50
MAPT P10636 4/20 0.50
HTT P42858 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
NFKB1 P19838 2/20 0.50
TP53 P04637 2/20 0.50
ALOX15 P16050 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxyquinoline SCHEMBL7261596 1.00 TSHR (0.81) TSHRMMP2CHRM1COMTADRA1A
Oxyquinoline SCHEMBL28194203 0.98 TSHR (0.78) TSHRMMP2CHRM1COMTADRA1A
Oxyquinoline SCHEMBL3070563 0.93 TSHR (0.70) TSHRMMP2CHRM1COMTADRA1A
Oxyquinoline SCHEMBL29100488 0.93 MMP2 (0.75) TSHRMMP2CHRM1COMTADRA1A
Oxyquinoline SCHEMBL29365411 0.90 TSHR (1.00) TSHRMMP2CHRM1COMTADRA1A
Oxyquinoline SCHEMBL29716519 0.90 TSHR (1.00) TSHRMMP2CHRM1COMTADRA1A
Oxyquinoline SCHEMBL37189 0.90 TSHR (1.00) TSHRMMP2CHRM1COMTADRA1A
Oxyquinoline SCHEMBL253313 0.90 TSHR (1.00) TSHRMMP2CHRM1COMTADRA1A
Oxyquinoline SCHEMBL15266589 0.90 MMP2 (0.70) TSHRMMP2CHRM1COMTADRA1A
Oxyquinoline SCHEMBL7187630 0.88 TSHR (0.88) TSHRMMP2CHRM1COMTADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107356742-B Method for rapidly detecting angiotensin I in batches 广州金域医学检验中心有限公司 2020-04-10 CN claimed
CN-107356742-A The method that rapid batch detects angiotensin I 广州金域医学检验中心有限公司 2017-11-17 CN claimed
WO-2009140215-A2 METHOD FOR TREATING DRUG-RESISTANT BACTERIAL AND OTHER INFECTIONS WITH CLIOQUINOL, PHANQUINONE, AND RELATED COMPOUNDS GERAGHTY, ERIN (US) 2009-11-19 WO claimed
CN-118956200-A PO43-8-OQ intercalated zinc-aluminum hydrotalcite and PO43-Preparation method of 8-OQ intercalated zinc-aluminum hydrotalcite flame-retardant epoxy acrylic acid coating and coating thereof 莆田学院 2024-11-15 CN disclosed
US-10959937-B2 Oil-in-water type organopolysiloxane emulsion and method for producing same, cosmetic raw material, and cosmetic product DOW TORAY CO., LTD. (JP) 2021-03-30 US disclosed
CN-107356742-B Method for rapidly detecting angiotensin I in batches 广州金域医学检验中心有限公司 2020-04-10 CN disclosed
US-20180280283-A1 OIL-IN-WATER TYPE ORGANOPOLYSILOXANE EMULSION AND METHOD FOR PRODUCING SAME, COSMETIC RAW MATERIAL, AND COSMETIC PRODUCT DOW TORAY CO., LTD. (JP) 2018-10-04 US disclosed
CN-107356742-A The method that rapid batch detects angiotensin I 广州金域医学检验中心有限公司 2017-11-17 CN disclosed
CN-105440348-A Phosphatized butadiene rubber material and preparation method thereof HEFEI JIEMING NEW MATERIAL TECH CO LTD 2016-03-30 CN disclosed
EP-1541633-B1 AQUEOUS SUSPENSION OF CROSSLINKED SILICONE PARTICLES, AQUEOUS EMULSION OF OIL CONTAINING CROSSLINKED SILICONE PARTICLES, AND COSMETIC INGREDIENTS DOW CORNING TORAY CO LTD (JP) 2013-01-16 EP disclosed
EP-1381651-B1 POLYORGANOSILOXANE EMULSION COMPOSITION AND A COSMETIC MATERIAL MADE THEREFROM DOW CORNING TORAY CO LTD (JP) 2011-06-29 EP disclosed
EP-1541633-A1 AQUEOUS SUSPENSION OF CROSSLINKED SILICONE PARTICLES, AQUEOUS EMULSION OF OIL CONTAINING CROSSLINKED SILICONE PARTICLES, AND COSMETIC INGREDIENTS Dow Corning Toray Silicone Company, Ltd. (JP) 2005-06-15 EP disclosed
US-20040147647-A1 Polyorganosiloxane micro-emulsion composition and raw material for cosmetics DOW CORNING TORAY SILICONE CO., LTD. (JP) 2004-07-29 US disclosed
US-20040138373-A1 Polyorganosiloxane emulsion composition and a cosmetic material made therefrom DOW TORAY CO., LTD. (JP) 2004-07-15 US disclosed
US-20040091438-A1 Polyorganosiloxane emulsions,process for producing the same and material for cosmetic preparation DOW CORNING TORAY SILICONE CO. LTD. (JP) 2004-05-13 US disclosed
EP-1406575-A2 POLYORGANOSILOXANE MICRO-EMULSION COMPOSITION AND RAW MATERIAL FOR COSMETICS Dow Corning Toray Silicone Co.,Ltd. Patent Department (JP) 2004-04-14 EP disclosed
EP-1394215-A1 POLYORGANOSILOXANE EMULSION, PROCESS FOR PRODUCING THE SAME, AND MATERIAL FOR COSMETIC PREPARATION Dow Corning Toray Silicone Co., Ltd. (JP) 2004-03-03 EP disclosed
EP-1381651-A1 POLYORGANOSILOXANE EMULSION COMPOSITION AND A COSMETIC MATERIAL MADE THEREFROM Dow Corning Toray Silicone Co.,Ltd. Patent Department (JP) 2004-01-21 EP disclosed
WO-2002094213-A2 POLYORGANOSILOXANE MICRO-EMULSION COMPOSITION AND RAW MATERIAL FOR COSMETICS DOW CORNING TORAY SILICONE CO.,LTD. (JP) 2002-11-28 WO disclosed
WO-2002088253-A1 POLYORGANOSILOXANE EMULSION COMPOSITION AND A COSMETIC MATERIAL MADE THEREFROM DOW CORNING TORAY SILICONE CO., LTD. (JP) 2002-11-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040091438-A1 Polyorganosiloxane emulsions,process for producing the same and material for cosmetic preparation CUTA, UNG, PCNA ADRA1A 1150/4885KDR 3530/4885TSHR 4487/4885
US-20040147647-A1 Polyorganosiloxane micro-emulsion composition and raw material for cosmetics UNG, PHOSPHO1, TPMT ADRA1A 1129/4885KDR 3791/4885TSHR 3740/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.