SCHEMBL2043071

SCHEMBL2043071

CC(C)CCc1cc2cc(F)cnc2n1S(=O)(=O)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PPARG P37231 5/20 0.38
PPARA Q07869 5/20 0.38
PPARD Q03181 2/20 0.36
TLR7 Q9NYK1 1/20 0.34
ALDH3A1 P30838 1/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
PTGDR Q13258 1/20 0.34
APLNR P35414 4/20 0.33
RECQL P46063 1/20 0.33
CACNA1G O43497 1/20 0.32
CACNA1H O95180 1/20 0.32
KCNH2 Q12809 1/20 0.32
TSHR P16473 1/20 0.32
NOD1 Q9Y239 2/20 0.32
CXCL8 P10145 1/20 0.32
PKM P14618 1/20 0.32
HTR6 P50406 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1963085 0.79 RECQL (0.39) PPARGPPARAALDH3A1PTGDR2PTGDR
SCHEMBL1959066 0.78 ALDH1A1 (0.39) PPARGPPARAALDH3A1PTGDR2PTGDR
SCHEMBL4197377 0.72 GRIN1 (0.39) PTGDR2PTGDRTSHRHTR6
SCHEMBL25153267 0.71 ENPP3 (0.44) PPARGPPARAPPARDPTGDR2TSHR
SCHEMBL30280436 0.71 ENPP3 (0.44) PPARGPPARAPPARDPTGDR2TSHR
SCHEMBL1963563 0.70 RECQL (0.36) RECQLHTR6
SCHEMBL1960448 0.70 RECQL (0.41) ALDH3A1PTGDR2PTGDRRECQLTSHR
SCHEMBL9701252 0.69 CYP2C19 (0.49) PPARGPPARAPPARDPTGDR2RECQL
SCHEMBL23246934 0.69 PIK3C3 (0.41) PPARGPPARAPPARDPTGDR2RECQL
SCHEMBL1962367 0.69 PTGS2 (0.40) ALDH3A1PTGDR2NOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513103-A1 AZAINDOLE GLUCOKINASE ACTIVATORS F. Hoffmann-La Roche AG (CH) 2012-10-24 EP disclosed
WO-2011073117-A1 AZAINDOLE GLUCOKINASE ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-23 WO disclosed