SCHEMBL20482159

SCHEMBL20482159

O=C(c1cc(F)cc(F)c1)[C@H]1CCCN1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.43
ALOX12 P18054 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 2/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20482718 1.00 THRB (0.43) THRBALOX12KMT2AALDH1A1CES2
SCHEMBL20482089 0.86 CES2 (0.39) THRBALOX12KMT2AALDH1A1CES2
SCHEMBL3532138 0.86 TAS1R3 (0.44) THRBALOX12KMT2A
SCHEMBL3532143 0.86 TAS1R3 (0.44) THRBALOX12KMT2A
SCHEMBL5339926 0.81 TDP1 (0.48)
SCHEMBL10132456 0.79 NPC1 (0.52) KMT2AALDH1A1
SCHEMBL20482125 0.79 KDM2B (0.52) KMT2AALDH1A1
SCHEMBL20482103 0.79 KDM2B (0.52) KMT2AALDH1A1
SCHEMBL20482097 0.79 ALDH1A1 (0.49) ALDH1A1
SCHEMBL3001673 0.79 ALDH1A1 (0.49) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018153820-A1 PROCESS FOR THE PREPARATION OF CHIRAL PYROLLIDINE-2-YL- METHANOL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2018-08-30 WO disclosed