SCHEMBL2053486

SCHEMBL2053486

Cc1[c]cccc1-c1ccc(F)cc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.35
GPR3 P46089 1/20 0.34
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 2/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34
ALOX12 P18054 1/20 0.34
ALDH1A1 P00352 3/20 0.33
MEN1 O00255 2/20 0.33
HPGD P15428 2/20 0.33
KMT2A Q03164 2/20 0.33
THRB P10828 1/20 0.33
HSD11B1 P28845 1/20 0.33
ACHE P22303 1/20 0.32
HSD17B1 P14061 1/20 0.32
HSD17B2 P37059 1/20 0.32
DPP4 P27487 1/20 0.32
TTR P02766 2/20 0.32
AKT1 P31749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2049820 0.86 PTPN1 (0.38) GPR3KDM4EHSD17B10POLBMAPT
SCHEMBL5868331 0.83 HSD11B1 (0.48) MAPK14GPR3MEN1KMT2AHSD11B1
SCHEMBL436195 0.81 GPR3 (0.36) MAPK14GPR3KDM4EHSD17B10ALDH1A1
SCHEMBL2015542 0.81 ACHE (0.39) KDM4EALDH1A1MEN1KMT2AHSD11B1
SCHEMBL15637654 0.79 PIK3R1 (0.37) MAPK14GPR3KDM4EHSD17B10ALDH1A1
SCHEMBL432712 0.79 MAPK14 (0.35) MAPK14GPR3KDM4EHSD17B10ALDH1A1
SCHEMBL17514930 0.78 MAPK14 (0.37) MAPK14GPR3HSD17B10ALDH1A1MEN1
SCHEMBL22115865 0.78
SCHEMBL2050049 0.77 MAPK14 (0.34) MAPK14KDM4EHSD17B10POLBMAPT
SCHEMBL2053315 0.76 PDK2 (0.35) MAPK14GPR3ALDH1A1HSD11B1PIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed