SCHEMBL2053580

SCHEMBL2053580

Cc1c[c]ccc1-c1cccc(F)c1F

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.35
ACHE P22303 1/20 0.34
DYRK1A Q13627 3/20 0.34
GAA P10253 2/20 0.33
MGAM O43451 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
BCAT1 P54687 1/20 0.33
CCNE2 O96020 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
MBNL1 Q9NR56 1/20 0.33
WDR5 P61964 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SLC9A1 P19634 1/20 0.30
KIF11 P52732 1/20 0.30
CTSA P10619 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012045 0.85 ACHE (0.41) ACHEGAAMGAMSIMGAM2
SCHEMBL8131456 0.83 BCAT1 (0.36) HSD11B1DYRK1ABCAT1CCNE2CCNE1
SCHEMBL2050739 0.81 ACHE (0.37) ACHE
SCHEMBL16720156 0.79 BCAT1 (0.33) BCAT1CCNE2CCNE1CDK2SLC9A1
SCHEMBL2014556 0.79 BCAT1 (0.33) BCAT1CCNE2CCNE1CDK2
SCHEMBL8122809 0.78 PDE2A (0.38) ACHENPC1CTSA
SCHEMBL14480559 0.78
SCHEMBL1371322 0.77 TSHR (0.39) ACHEGAANPC1RAB9ASMN1; SMN2
SCHEMBL2049472 0.76 HSD11B1 (0.42) HSD11B1BCAT1CCNE2CCNE1CDK2
SCHEMBL5673742 0.75 CYP1A2 (0.33) BCAT1CCNE2CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed