SCHEMBL2058331

SCHEMBL2058331

O=C(O)c1ccccc1NC(=O)c1ccccc1C(=O)O

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.68
KMT2A Q03164 6/20 0.68
MEN1 O00255 3/20 0.68
PKM P14618 1/20 0.68
DHODH Q02127 1/20 0.66
NPSR1 Q6W5P4 2/20 0.61
PRNP P04156 1/20 0.61
PPARG P37231 1/20 0.61
RXFP1 Q9HBX9 1/20 0.61
NCOR2 Q9Y618 1/20 0.61
NPC1 O15118 3/20 0.58
RAB9A P51151 3/20 0.58
HPGD P15428 2/20 0.58
CA12 O43570 1/20 0.58
CA2 P00918 1/20 0.58
CA9 Q16790 1/20 0.58
ALOX15 P16050 1/20 0.58
POLB P06746 1/20 0.58
TP53 P04637 1/20 0.57
CYP1A2 P05177 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10481401 0.89 KMT2A (0.60) ALDH1A1KMT2AMEN1PKMDHODH
SCHEMBL14398957 0.89 NPSR1 (0.63) ALDH1A1KMT2AMEN1PKMDHODH
SCHEMBL14398138 0.89 NPSR1 (0.68) ALDH1A1KMT2AMEN1PKMDHODH
SCHEMBL11284668 0.89 PDCD1 (0.64) ALDH1A1KMT2AMEN1PKMDHODH
SCHEMBL328588 0.89 ALDH1A1 (0.82) ALDH1A1KMT2AMEN1PKMNPSR1
SCHEMBL14087662 0.87 DHODH (0.69) ALDH1A1KMT2AMEN1PKMDHODH
SCHEMBL4669122 0.86 LMNA (0.76) ALDH1A1KMT2AMEN1PKMDHODH
SCHEMBL11405554 0.86 LMNA (0.76) ALDH1A1KMT2AMEN1PKMDHODH
SCHEMBL15183709 0.86 KMT2A (0.77) KMT2AMEN1PKMDHODHPPARG
SCHEMBL28965115 0.86 LMNA (0.76) ALDH1A1KMT2AMEN1PKMNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2115111-B1 BENZOPHENONE OR BENZOIC ACID ANILIDE DERIVATIVES CONTAINING CARBOXYL GROUPS AS ENZYME STABILIZERS HENKEL AG & CO KGAA (DE) 2014-04-30 EP claimed
US-7968508-B2 Benzophenone or benzoic acid anilide derivatives containing carboxyl groups as enzyme stabilizers HENKEL AG & CO. KGAA (DE) 2011-06-28 US claimed
US-20100062964-A1 Benzophenone or Benzoic Acid Anilide Derivatives containing Carboxyl Groups as Enzyme Stabilizers HENKEL AG & CO., KGAA (DE) 2010-03-11 US claimed
EP-0172890-A4 ACCUMULATED THERMAL EXPOSURE RESPONDER AND METHOD OF USE. CONTROLLED CHEMICALS INC (US) 1989-07-25 EP claimed
EP-0172890-A1 ACCUMULATED THERMAL EXPOSURE RESPONDER AND METHOD OF USE CONTROLLED CHEMICALS INCORPORATED (US) 1986-03-05 EP claimed
WO-1985003775-A1 ACCUMULATED THERMAL EXPOSURE RESPONDER AND METHOD OF USE CONTROLLED CHEMICALS INCORPORATED (US) 1985-08-29 WO claimed
US-4533640-A INDICATING DETERIORATION OF PERISHABLE GOODS CONTROLLED CHEMICALS INCORPORATED A MI CORP 1985-08-06 US claimed
JP-55133425-A None JP disclosed
US-11045476-B2 Compounds and methods for inducing chondrogenesis THE SCRIPPS RESEARCH INSTITUTE (US) 2021-06-29 US disclosed
US-20200188407-A1 COMPOUNDS AND METHODS FOR INDUCING CHONDROGENESIS THE SCRIPPS RESEARCH INSTITUTE 2020-06-18 US disclosed
US-10166237-B2 Compounds and methods for inducing chondrogenesis THE SCRIPPS RESEARCH INSTITUTE (US) 2019-01-01 US disclosed
US-20170112843-A1 COMPOUNDS AND METHODS FOR INDUCING CHONDROGENESIS THE SCRIPPS RESEARCH INSTITUTE 2017-04-27 US disclosed
US-9464065-B2 Compounds and methods for inducing chondrogenesis THE SCRIPPS RESEARCH INSTITUTE (US) 2016-10-11 US disclosed
WO-1994025501-A1 EPOXY RESINS CONTAINING THIADIAZOLE AND/OR OXADIAZOLE MOIETIES THE DOW CHEMICAL COMPANY (US) 1994-11-10 WO disclosed
EP-0172890-A4 ACCUMULATED THERMAL EXPOSURE RESPONDER AND METHOD OF USE. CONTROLLED CHEMICALS INC (US) 1989-07-25 EP disclosed
US-4795714-A MONITOR OF THERMAL EXPOSURE WHICH SIGNALS DETERIORATION OF PERSHIBLE GOODS SHAFER JULES A (US) 1989-01-03 US disclosed
EP-0172890-A1 ACCUMULATED THERMAL EXPOSURE RESPONDER AND METHOD OF USE CONTROLLED CHEMICALS INCORPORATED (US) 1986-03-05 EP disclosed
WO-1985003775-A1 ACCUMULATED THERMAL EXPOSURE RESPONDER AND METHOD OF USE CONTROLLED CHEMICALS INCORPORATED (US) 1985-08-29 WO disclosed
US-4533640-A INDICATING DETERIORATION OF PERISHABLE GOODS CONTROLLED CHEMICALS INCORPORATED A MI CORP 1985-08-06 US disclosed
JP-S55133425-A PREPARATION OF AMIDE GROUP-CONTAINING POLYESTER COPOLYMER TORAY IND INC 1980-10-17 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10166237-B2 Compounds and methods for inducing chondrogenesis COL2A1, BMP4, BMP2 ALDH1A1 63/4885KMT2A 3000/4885MEN1 4660/4885
US-11045476-B2 Compounds and methods for inducing chondrogenesis COL2A1, BMP4, COL1A1 ALDH1A1 52/4885KMT2A 3871/4885MEN1 4679/4885
US-20170112843-A1 COMPOUNDS AND METHODS FOR INDUCING CHONDROGENESIS COL2A1, BMP4, BMP2 ALDH1A1 63/4885KMT2A 3000/4885MEN1 4660/4885
US-20200188407-A1 COMPOUNDS AND METHODS FOR INDUCING CHONDROGENESIS COL2A1, BMP4, COL1A1 ALDH1A1 52/4885KMT2A 3871/4885MEN1 4679/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.