SCHEMBL20620649

SCHEMBL20620649

c1ccc(-c2ccc(-c3cc(N(c4ccccc4)c4ccc(-c5ccccc5)cc4)ccc3-c3ccc(-c4ccc(N(c5ccccc5)c5ccc(-c6ccccc6)cc5)cc4)cc3)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 4/20 0.43
ALDH1A1 P00352 4/20 0.43
MAPT P10636 3/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
ATM Q13315 2/20 0.37
NPC1 O15118 2/20 0.37
LMNA P02545 2/20 0.37
HTT P42858 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
CRHBP P24387 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20620409 1.00 L3MBTL1 (0.43) L3MBTL1ALDH1A1MAPTKDM4ECYP1A2
SCHEMBL2604758 1.00 L3MBTL1 (0.43) L3MBTL1ALDH1A1MAPTKDM4ECYP1A2
SCHEMBL20620705 1.00 L3MBTL1 (0.43) L3MBTL1ALDH1A1MAPTKDM4ECYP1A2
SCHEMBL20558789 1.00 L3MBTL1 (0.43) L3MBTL1ALDH1A1MAPTKDM4ECYP1A2
SCHEMBL20620655 1.00 L3MBTL1 (0.43) L3MBTL1ALDH1A1MAPTKDM4ECYP1A2
SCHEMBL24079326 1.00 L3MBTL1 (0.43) L3MBTL1ALDH1A1MAPTKDM4ECYP1A2
SCHEMBL20582563 1.00 L3MBTL1 (0.43) L3MBTL1ALDH1A1MAPTKDM4ECYP1A2
SCHEMBL20484377 1.00 L3MBTL1 (0.43) L3MBTL1ALDH1A1MAPTKDM4ECYP1A2
SCHEMBL20484439 1.00 L3MBTL1 (0.43) L3MBTL1ALDH1A1MAPTKDM4ECYP1A2
SCHEMBL17780076 1.00 L3MBTL1 (0.43) L3MBTL1ALDH1A1MAPTKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230284515-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANIC LIGHT-EMITTING ELEMENT USING THE SAME SFC CO., LTD. (KR) 2023-09-07 US disclosed
US-20230284515-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANIC LIGHT-EMITTING ELEMENT USING THE SAME SFC CO., LTD. (KR) 2023-09-07 US disclosed
EP-3750971-B1 ORGANIC ELECTROLUMINESCENT DEVICE SFC CO LTD (KR) 2023-02-22 EP disclosed
US-20220102635-A1 ORGANIC LIGHT-EMITTING ELEMENT USING POLYCYCLIC AROMATIC DERIVATIVE COMPOUND SFC CO., LTD. (KR) 2022-03-31 US disclosed
EP-3889236-A1 ORGANIC LIGHT-EMITTING ELEMENT USING POLYCYCLIC AROMATIC DERIVATIVE COMPOUND SFC Co., Ltd. (KR) 2021-10-06 EP disclosed
US-20210167293-A1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME SFC CO., LTD. (KR) 2021-06-03 US disclosed
EP-3660024-B1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME SFC CO LTD (KR) 2021-05-05 EP disclosed
US-10981938-B2 Polycyclic aromatic compounds and organic electroluminescent devices using the same SFC CO., LTD. (KR) 2021-04-20 US disclosed
US-20200395553-A1 ORGANIC ELECTROLUMINESCENT DEVICE SFC CO., LTD. (KR) 2020-12-17 US disclosed
EP-3750971-A1 ORGANIC ELECTROLUMINESCENT DEVICE SFC Co., Ltd. (KR) 2020-12-16 EP disclosed
US-20200172558-A1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME SFC CO., LTD. (KR) 2020-06-04 US disclosed
EP-3660024-A1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME SFC Co., Ltd. (KR) 2020-06-03 EP disclosed
US-20200161552-A1 INDOLOCARBAZOLE DERIVATIVES AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME SFC CO., LTD. (KR) 2020-05-21 US disclosed
US-20190006596-A1 ORGANIC ELECTROLUMINESCENT DEVICE HODOGAYA CHEMICAL CO., LTD. (JP) 2019-01-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200172558-A1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME DDC, TYR, DDT L3MBTL1 2066/4885ALDH1A1 711/4885MAPT 1909/4885
US-20220102635-A1 ORGANIC LIGHT-EMITTING ELEMENT USING POLYCYCLIC AROMATIC DERIVATIVE COMPOUND TRPA1, TYR, ZKSCAN2 L3MBTL1 508/4885ALDH1A1 1979/4885MAPT 223/4885
US-20230284515-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANIC LIGHT-EMITTING ELEMENT USING THE SAME ARNT, AHR, TYR L3MBTL1 429/4885ALDH1A1 605/4885MAPT 209/4885
US-20190006596-A1 ORGANIC ELECTROLUMINESCENT DEVICE SLC43A1, SLC7A5, SLCO4C1 L3MBTL1 634/4885ALDH1A1 227/4885MAPT 1328/4885
US-20210167293-A1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME DDC, TYR, DDT L3MBTL1 2066/4885ALDH1A1 711/4885MAPT 1909/4885
US-10981938-B2 Polycyclic aromatic compounds and organic electroluminescent devices using the same DDC, TYR, DDT L3MBTL1 2066/4885ALDH1A1 711/4885MAPT 1909/4885
US-20200395553-A1 ORGANIC ELECTROLUMINESCENT DEVICE LEF1, AP2A2, CCNA1 L3MBTL1 821/4885ALDH1A1 17/4885MAPT 2312/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.