SCHEMBL2069110

SCHEMBL2069110

O=C(Nc1ccccc1)c1c(O)c2ccccc2[nH]c1=O

nearest known ligand 0.78

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 10/20 0.78
MEN1 O00255 8/20 0.78
NPC1 O15118 7/20 0.78
RAB9A P51151 7/20 0.78
EGFR P00533 1/20 0.74
L3MBTL1 Q9Y468 1/20 0.70
RXFP1 Q9HBX9 1/20 0.67
SERPINE1 P05121 1/20 0.65
KDM4E B2RXH2 7/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
NLRP3 Q96P20 1/20 0.64
MAPT P10636 3/20 0.63
POLB P06746 1/20 0.63
PKM P14618 1/20 0.62
ALDH1A1 P00352 2/20 0.61
GAA P10253 1/20 0.61
NPSR1 Q6W5P4 2/20 0.61
HTT P42858 1/20 0.61
LMNA P02545 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3982130 0.92 KMT2A (0.67) KMT2AMEN1NPC1RAB9AEGFR
SCHEMBL2815751 0.92 KMT2A (0.74) KMT2AMEN1NPC1RAB9AEGFR
SCHEMBL14311488 0.89 RAB9A (0.76) KMT2AMEN1NPC1RAB9AEGFR
SCHEMBL2299556 0.89 KMT2A (0.67) KMT2AMEN1NPC1RAB9AEGFR
SCHEMBL13598030 0.89 KMT2A (0.67) KMT2AMEN1NPC1RAB9AEGFR
SCHEMBL13597992 0.88 SERPINE1 (0.69) KMT2AMEN1NPC1RAB9AEGFR
SCHEMBL14311489 0.86 RAB9A (1.00) KMT2AMEN1NPC1RAB9AEGFR
SCHEMBL13598036 0.86 KMT2A (0.78) KMT2AMEN1NPC1RAB9AEGFR
SCHEMBL13597991 0.86 KMT2A (0.67) KMT2AMEN1NPC1RAB9AEGFR
SCHEMBL13598024 0.85 KMT2A (0.73) KMT2AMEN1NPC1RAB9AEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230202982-A1 5-CHLORO-4-HYDROXY-1-METHYL-2-OXO-N-PHENYL-QUINOLINE-3-CARBOXAMIDE POTASSIUM SALT FOR TREATING INFLAMMATORY BOWEL DISEASES AQILION AB (SE) 2023-06-29 US disclosed
US-20230167064-A1 TREATMENTS OF INFLAMMATORY BOWEL DISEASE AQILION AB (SE) 2023-06-01 US disclosed
CN-115916200-A Treatment of inflammatory bowel disease 阿奎利恩有限公司 2023-04-04 CN disclosed
EP-4142724-A1 TREATMENTS OF INFLAMMATORY BOWEL DISEASE Aqilion AB (SE) 2023-03-08 EP disclosed
US-20220031628-A1 NANOPARTICLES FOR PREPARING REGULATORY B CELLS UNIVERSITÉ PARIS CITÉ (FR) 2022-02-03 US disclosed
WO-2021219879-A1 TREATMENTS OF INFLAMMATORY BOWEL DISEASE AQILION AB (SE) 2021-11-04 WO disclosed
US-20210220481-A1 BIOCOMPATIBLE TOLEROGENIC NANOPARTICLES UNIVERSITÉ PARIS CITÉ (FR) 2021-07-22 US disclosed
EP-3829557-A1 BIOCOMPATIBLE TOLEROGENIC NANOPARTICLES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2021-06-09 EP disclosed
WO-2020025408-A1 BIOCOMPATIBLE TOLEROGENIC NANOPARTICLES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2020-02-06 WO disclosed
US-20180071376-A1 TOLEROGENIC NANOPARTICLES FOR TREATING DIABETES MELLITUS THE BRIGHAM AND WOMEN'S HOSPITAL, INC. 2018-03-15 US disclosed
EP-2627638-A1 1,2-DIHYDRO-4-HYDROXY-2-OXO-QUINOLINE-3-CARBOXANILIDES AS AHR ACTIVATORS. Immunahr AB (SE) 2013-08-21 EP disclosed
US-20130203703-A1 1,2-DIHYDRO-4-HYDROXY-2-OXO-QUINOLINE-3-CARBOXANILIDES AS AHR ACTIVATORS IMMUNAHR AB (SE) 2013-08-08 US disclosed
US-20130203703-A1 1,2-DIHYDRO-4-HYDROXY-2-OXO-QUINOLINE-3-CARBOXANILIDES AS AHR ACTIVATORS IMMUNAHR AB (SE) 2013-08-08 US disclosed
CN-103153959-A 1,2-dihydro-4-hydroxy-2-oxo-quinoline-3-carboxanilides as ahr activators IMMUNAHR AB 2013-06-12 CN disclosed
CN-103153959-A 1,2-dihydro-4-hydroxy-2-oxo-quinoline-3-carboxanilides as ahr activators IMMUNAHR AB 2013-06-12 CN disclosed
CN-103153959-A 1,2-dihydro-4-hydroxy-2-oxo-quinoline-3-carboxanilides as ahr activators IMMUNAHR AB 2013-06-12 CN disclosed
WO-2012050500-A1 1,2-DIHYDRO-4-HYDROXY-2-OXO-QUINOLINE-3-CARBOXANILIDES AS AHR ACTIVATORS. PETTERSSON LARS (SE) 2012-04-19 WO disclosed
WO-2012050500-A1 1,2-DIHYDRO-4-HYDROXY-2-OXO-QUINOLINE-3-CARBOXANILIDES AS AHR ACTIVATORS. PETTERSSON LARS (SE) 2012-04-19 WO disclosed
US-20090325948-A1 INHIBITORS OF UNDECAPRENYL PYROPHOSPHATE SYNTHASE HURLEY TIMOTHY BRIAN 2009-12-31 US disclosed
US-20090325948-A1 INHIBITORS OF UNDECAPRENYL PYROPHOSPHATE SYNTHASE HURLEY TIMOTHY BRIAN 2009-12-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090325948-A1 INHIBITORS OF UNDECAPRENYL PYROPHOSPHATE SYNTHASE FDPS, UMPS, GGPS1 KMT2A 4780/4885MEN1 2345/4885NPC1 163/4885
US-20210220481-A1 BIOCOMPATIBLE TOLEROGENIC NANOPARTICLES IAPP, AHR, ARNT KMT2A 3166/4885MEN1 2413/4885NPC1 1415/4885
US-20220031628-A1 NANOPARTICLES FOR PREPARING REGULATORY B CELLS IAPP, IL2, CCR10 KMT2A 2962/4885MEN1 2738/4885NPC1 1843/4885
US-20180071376-A1 TOLEROGENIC NANOPARTICLES FOR TREATING DIABETES MELLITUS IAPP, NFATC1, CD4 KMT2A 3866/4885MEN1 4304/4885NPC1 1204/4885
US-20230167064-A1 TREATMENTS OF INFLAMMATORY BOWEL DISEASE SLC10A2, SI, ALPI KMT2A 3547/4885MEN1 2883/4885NPC1 504/4885
US-20130203703-A1 1,2-DIHYDRO-4-HYDROXY-2-OXO-QUINOLINE-3-CARBOXANILIDES AS AHR ACTIVATORS AHR, HRH4, ARNT KMT2A 761/4885MEN1 3486/4885NPC1 3628/4885
US-20230202982-A1 5-CHLORO-4-HYDROXY-1-METHYL-2-OXO-N-PHENYL-QUINOLINE-3-CARBOXAMIDE POTASSIUM SALT FOR TREATING INFLAMMATORY BOWEL DISEASES SLC10A2, KCNK5, KCNQ5 KMT2A 88/4885MEN1 2958/4885NPC1 357/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.