SCHEMBL206956

SCHEMBL206956

COc1ccc(N2CCN(C(=O)CCCC(=O)NC3CCC(Cc4ccccc4)(N(C)C)CC3)CC2)c(OC)c1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 2/20 0.43
DRD2 P14416 1/20 0.43
SIGMAR1 Q99720 2/20 0.43
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HTR7 P34969 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206125 0.88 ADAMTS4 (0.47) SIGMAR1MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL207058 0.86 SIGMAR1 (0.55) SIGMAR1MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL205294 0.84 AR (0.56) DRD2HTR7MEN1KMT2ASMN1; SMN2
SCHEMBL206937 0.83 MTNR1B (0.49) SIGMAR1ALDH1A1GAA
SCHEMBL205791 0.82 MAPT (0.52) MEN1KMT2ASMN1; SMN2ALDH1A1LMNA
SCHEMBL207857 0.80 LMNA (0.55) HTR7KMT2ALMNAMAPTGAA
SCHEMBL206177 0.78 ALDH1A1 (0.48) KMT2AALDH1A1GAA
SCHEMBL206079 0.78 OPRM1 (0.54) SIGMAR1
SCHEMBL207144 0.77 ADAMTS4 (0.47) DRD4SIGMAR1MEN1KMT2ALMNA
SCHEMBL4075869 0.77 ALDH1A1 (0.57) HTR7MEN1KMT2ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088763-B2 e.g. N-[1-(2,6-dichloro-benzyl)-pyrrolidin-3-yl]-N'-[4-dimethylamino-4-(4-methyl-benzyl)-cyclohexyl]-succinamide; noradrenaline and serotonin reuptake ihibitor; opioid ORL-1 receptor ligand; analgesic, antidepressant, anxiolytic agent, neurodegenerative diseases GRUENENTHAL GMBH (DE) 2012-01-03 US claimed
US-8088763-B2 e.g. N-[1-(2,6-dichloro-benzyl)-pyrrolidin-3-yl]-N'-[4-dimethylamino-4-(4-methyl-benzyl)-cyclohexyl]-succinamide; noradrenaline and serotonin reuptake ihibitor; opioid ORL-1 receptor ligand; analgesic, antidepressant, anxiolytic agent, neurodegenerative diseases GRUENENTHAL GMBH (DE) 2012-01-03 US disclosed