SCHEMBL20726382

SCHEMBL20726382

C/C(O)=C1\C(=O)Nc2cc(O)c(-c3ccc(C#N)cc3)cc21

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.48
CHEK1 O14757 3/20 0.39
MDM2 Q00987 3/20 0.39
WEE1 P30291 1/20 0.38
LRRK2 Q5S007 1/20 0.35
MMP3 P08254 1/20 0.35
KDM1A O60341 1/20 0.34
MAOA P21397 1/20 0.34
TOP2A P11388 1/20 0.34
TOP2B Q02880 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ATM Q13315 1/20 0.34
KDR P35968 1/20 0.34
AR P10275 1/20 0.34
PAK4 O96013 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20726381 0.81 PGR (0.43) EGFRLRRK2ALDH1A1KDRAR
SCHEMBL20726502 0.77 BRD4 (0.39) EGFRCHEK1MAOAALDH1A1KDR
SCHEMBL20726357 0.76 BRD4 (0.40) EGFRCHEK1ALDH1A1
SCHEMBL20726412 0.75 PRKDC (0.43) CHEK1
SCHEMBL20726495 0.75 EGFR (0.35) EGFRCHEK1KDR
SCHEMBL20726384 0.71 PDE3B (0.50) EGFRKDR
SCHEMBL20726441 0.71 EGFR (0.40) EGFRKDR
SCHEMBL20726427 0.70 BRD4 (0.42) EGFRCHEK1MAOAKDR
SCHEMBL20726393 0.69 EGFR (0.39) EGFRCHEK1KDR
SCHEMBL20726451 0.69 EGFR (0.39) EGFRCHEK1WEE1LRRK2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3083611-B1 OXINDOLE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE IN THE TREATMENT OF AMPK-RELATED DISEASES SANOFI SA (FR) 2019-02-13 EP disclosed